Year: 2025
Design, synthesis, in silico and in vitro evaluation of pyrrole-indole hybrids as dual tubulin and aromatase inhibitors with potent anticancer activities
Rsc Advances, 2025-06-27, Vol. 15 (27)
Year: 2024
Synthesis, in silico, in vitro evaluation of furanyl- and thiophenyl-3-phenyl-1H-indole-2-carbohydrazide derivatives as tubulin inhibitors and anticancer agents
Rsc Medicinal Chemistry, 2024-05-28, Vol. 15 (7)
Metal- and photocatalyst-free approach to visible-light-induced acylation of quinoxalinones
Organic and Biomolecular Chemistry, 2024-04-30, Vol. 22 (29)
A structure-based virtual high-throughput screening, molecular docking, molecular dynamics and MM/PBSA study identified novel putative drug-like dual inhibitors of trypanosomal cruzain and rhodesain cysteine proteases
Molecular Diversity, 2024-04-01, Vol. 28 (2)
Year: 2022
Discovery of potent antiproliferative agents from selected oxygen heterocycles as EGFR tyrosine kinase inhibitors from the U.S. National Cancer Institute database by in silico screening and bioactivity evaluation
Bioorganic and Medicinal Chemistry Letters, 2022-02-15, Vol. 58
OXIDATIVE FRAGMENTATION OF CYTISINE AS AN ENTRY TO THE BIS(PIPERIDINE) SCAFFOLD OF VIRGIDIVARINE
Heterocycles, 2022-01-01, Vol. 105 (1)
Year: 2021
Visible-light-mediated decarboxylative alkylation of 2-pyridone derivatives: Via a C3-selective C-H functionalization
Organic and Biomolecular Chemistry, 2021-11-14, Vol. 19 (42)
In Silico-Guided Rational Drug Design and Semi-synthesis of C(2)-Functionalized Huperzine A Derivatives as Acetylcholinesterase Inhibitors
ACS Omega, 2021-08-03, Vol. 6 (30)
Identification of new 3-phenyl-1H-indole-2-carbohydrazide derivatives and their structure–activity relationships as potent tubulin inhibitors and anticancer agents: A combined in silico, in vitro and synthetic study
Bioorganic Chemistry, 2021-05-01, Vol. 110
Year: 2018
Iridium-Catalysed C-H Borylation of 2-Pyridones; Bisfunctionalisation of CC4
Synthesis Germany, 2018-06-29, Vol. 50 (17)
(-)-Cytisine: Access to a stereochemically defined and functionally flexible piperidine scaffold
Organic and Biomolecular Chemistry, 2018-01-01, Vol. 16 (32)
Year: 2017
Synthesis of Functionalized Alkenes by a Transition-Metal-Free Zweifel Coupling
Organic Letters, 2017-05-19, Vol. 19 (10)