RESEARCH IN CHEMICAL SCIENCES (CS)

2024

4-Aryl-1H-isochromenes Synthesis from Triol Derivatives through Brønsted Acid-Catalyzed Pinacol Rearrangement/Intramolecular Cyclization Sequence

By: Ieawsuwan, W., Limjirawatthana, S., Ploypradith, P., and Ruchirawat, S.

Asian Journal of Organic Chemistry
Vol.: 13
No.: 2
Page:
Published: 2024
doi: https://doi.org/10.1002/ajoc.202300578

Albiflorenes A–L, polyoxygenated cyclohex(a/e)ne diterpene esters from Kaempferia albiflora

By: Booranaseensuntorn, P., Boonsombat, J., Thongnest, S., Batsomboon, P., Reuk-Ngam, N., Khlaychan, P., Ruchisansakun, S., Kittakoop, P., Techasakul, S., Mahidol, C., and Ruchirawat, S.

Scientific Reports
Vol.: 14
No.: 1
Page:
Published: 2024
doi: https://doi.org/10.1038/s41598-024-64889-6

Altenusin, a fungal metabolite, alleviates TGF-β1-induced EMT in renal proximal tubular cells and renal fibrosis in unilateral ureteral obstruction

By: Thipboonchoo, N., Fongsupa, S., Sureram, S., Sa-nguansak, S., Kesornpun, C., Kittakoop, P., and Soodvilai, S.

Heliyon
Vol.: 10
No.: 3
Page:
Published: 2024
doi: https://doi.org/10.1016/j.heliyon.2024.e24983

Breast Cancer Prevention by Dietary Polyphenols: Microemulsion Formulation and In Vitro Studies

By: Cristy, G. P., Liana, D., Chatwichien, J., Aonbangkhen, C., Srisomsap, C., and Phanumartwiwath, A.

Scientia Pharmaceutica
Vol.: 92
No.: 2
Page:
Published: 2024
doi: https://doi.org/10.3390/scipharm92020025

Cascade Cyclization of o-(2-Acyl-1-ethynyl)benzaldehydes with Amino Acid Derivatives: Synthesis of Indeno[2,1-c]pyran-3-ones and 1-Oxazolonylisobenzofurans via the Erlenmeyer-Plöchl Azlactone Reaction

By: Worayuthakarn, R., Suddee, N., Theppitak, C., Chainok, K., Ruchirawat, S., and Thasana, N.

ACS Omega
Vol.: 9
No.: 36
Page: 37814-37842
Published: 2024
doi: https://doi.org/10.1021/acsomega.4c03842

Chemical constituents from Microstachys chamaelea (Euphorbiaceae) with cytotoxic and antioxidant properties

By: Sangsopha, W., Schevenels, F. T., Lekphrom, R., and Ruchirawat, S.

Natural Product Research
Vol.:
No.:
Page:
Published: 2024
doi: https://doi.org/10.1080/14786419.2024.2315598

Controllable Chemoselectivity Cascade Reactions for the Synthesis of Phenanthrenols via Palladium-Catalyzed-Suzuki/Heck Reaction and Michael Addition

By: Yongpanich, P., Chatrangsan, K., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.

Chemistry – An Asian Journal
Vol.: 19
No.: 9
Page:
Published: 2024
doi: https://doi.org/10.1002/asia.202400126

Cytotoxic stress caused by azalamellarin D (AzaD) interferes with cellular protein translation by targeting the nutrient-sensing kinase mTOR

By: Meerod, T., Sangsuwan, R., Klumthong, K., Chantrathonkul, B., Phutubtim, N., Govitrapong, P., Ruchirawat, S., Ploypradith, P., and Sopha, P.

Journal of Biochemistry
Vol.: 176
No.: 2
Page: 139-153
Published: 2024
doi: https://doi.org/10.1093/jb/mvae038

Dihydro-10H-indeno[1,2-b]benzofurans and Tetrahydroindeno[1,2-c]isochromenes via Stereoselective Intramolecular Carbocation Cascade Cyclization

By: Tangdenpaisal, K., Kheakwanwong, W., Ruchirawat, S., and Ploypradith, P.

Journal of Organic Chemistry
Vol.: 89
No.: 5
Page: 2964-2983
Published: 2024
doi: https://doi.org/10.1021/acs.joc.3c02380

Diphenyl ethers from the cultured lichen mycobiont of Graphis handelii Zahlbr

By: Tran, T. M. D., Aonbangkhen, C., Duong, T. H., Nguyen, T. H. M., Ho, M. T. T., Chavasiri, W., Wongsuwan, S., Chatwichien, J., Giao Vo, T. P., Nguyen, N. H., Kiriwan, D., and Choowongkomon, K.

Heliyon
Vol.: 10
No.: 4
Page:
Published: 2024
doi: https://doi.org/10.1016/j.heliyon.2024.e25763

Discovery of procyanidin condensed tannins of (−)-epicatechin from Kratom, Mitragyna speciosa, as virucidal agents against SARS-CoV-21

By: Sureram, S., Chutiwitoonchai, N., Pooprasert, T., Sangsopha, W., Limjiasahapong, S., Jariyasopit, N., Sirivatanauksorn, Y., Khoomrung, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.

International Journal of Biological Macromolecules
Vol.: 273
No.:
Page:
Published: 2024
doi: https://doi.org/10.1016/j.ijbiomac.2024.133059

Effects of barakol from Cassia siamea on neuroblastoma SH-SY5Y cell line: A potential combined therapy with doxorubicin

By: Wongsawatkul, O., Buachan, P., Jaisin, Y., Busarakumtragul, P., Chainakul, S., Watanapokasin, R., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.

Heliyon
Vol.: 10
No.: 3
Page:
Published: 2024
doi: https://doi.org/10.1016/j.heliyon.2024.e24694

Electron Donor-Acceptor Complex-Enabled Autoinductive Conversion of Acylnitromethanes to Acylnitrile Oxides in a Photochemical Machetti-De Sarlo Reaction: Synthesis of 5-Substituted 3-Acylisoxazoles

By: Arunkirirote, P., Suwalak, P., Chaisan, N., Tummatorn, J., Ruchirawat, S., and Thongsornkleeb, C.

Organic Letters
Vol.:
No.:
Page:
Published: 2024
doi: https://doi.org/10.1021/acs.orglett.4c02708

Enantioselective Reductive Cyclization of Alkynyl-Tethered Cyclohexadienones Catalyzed by Rhodium Complexes

By: Wang, Y. F., Wang, F., Yang, D. D., Kittakoop, P., Tan, Y. X., and Tian, P.

Organic Letters
Vol.: 26
No.: 27
Page: 5614-5619
Published: 2024
doi: https://doi.org/10.1021/acs.orglett.4c01276

Evolution-guided engineering of trans-acyltransferase polyketide synthases

By: Mabesoone, M. F. J., Leopold-Messer, S., Minas, H. A., Chepkirui, C., Chawengrum, P., Reiter, S., Meoded, R. A., Wolf, S., Genz, F., Magnus, N., Piechulla, B., Walker, A. S., and Piel, J.

Science
Vol.: 383
No.: 6689
Page: 1312-1317
Published: 2024
doi: https://doi.org/10.1126/science.adj7621

Facile metabolic reprogramming distinguishes mycobacterial adaptation to hypoxia and starvation: ketosis drives starvation-induced persistence in M. bovis BCG

By: Davis, N. K., Chionh, Y. H., McBee, M. E., Hia, F., Ma, D., Cui, L., Sharaf, M. L., Cai, W. M., Jumpathong, W., Levine, S. S., Alonso, S., and Dedon, P. C.

Communications Biology
Vol.: 7
No.: 1
Page:
Published: 2024
doi: https://doi.org/10.1038/s42003-024-06562-2

Grewiifopenes A–K, bioactive clerodane diterpenoids from Casearia grewiifolia Vent

By: Pailee, P., Batsomboon, P., Yaosanit, W., Thananthaisong, T., Mahidol, C., Ploypradith, P., Reuk-ngam, N., Khlaychan, P., Techasakul, S., Ruchirawat, S., and Prachyawarakorn, V.

Natural Products and Bioprospecting
Vol.: 14
No.: 1
Page:
Published: 2024
doi: https://doi.org/10.1007/s13659-024-00475-7

Huperzine A Regulates the Physiological Homeostasis of Amyloid Precursor Protein Proteolysis and Tau Protein Conformation—A Computational and Experimental Investigation

By: Wongjaikam, S., Nopparat, C., Boontem, P., Panmanee, J., Thasana, N., Shukla, M., and Govitrapong, P.

Biology
Vol.: 13
No.: 7
Page:
Published: 2024
doi: https://doi.org/10.3390/biology13070518

Inhibition of Giardia duodenalis by isocryptolepine -triazole adducts and derivatives

By: Popruk, S., Tummatorn, J., Sreesai, S., Ampawong, S., Thiangtrongjit, T., Tipthara, P., Tarning, J., Thongsornkleeb, C., Ruchirawat, S., and Reamtong, O.

International Journal for Parasitology: Drugs and Drug Resistance
Vol.: 26
No.:
Page:
Published: 2024
doi: https://doi.org/10.1016/j.ijpddr.2024.100561

Ligand-Based Virtual Screening for Discovery of Indole Derivatives as Potent DNA Gyrase ATPase Inhibitors Active against Mycobacterium tuberculosis and Hit Validation by Biological Assays

By: Pakamwong, B., Thongdee, P., Kamsri, B., Phusi, N., Taveepanich, S., Chayajarus, K., Kamsri, P., Punkvang, A., Hannongbua, S., Sangswan, J., Suttisintong, K., Sureram, S., Kittakoop, P., Hongmanee, P., Santanirand, P., Leanpolchareanchai, J., Spencer, J., Mulholland, A. J., and Pungpo, P.

Journal of Chemical Information and Modeling
Vol.: 64
No.: 15
Page: 5991-6002
Published: 2024
doi: https://doi.org/10.1021/acs.jcim.4c00511

Metal- and photocatalyst-free approach to visible-light-induced acylation of quinoxalinones

By: Niwetmarin, W., Saesian, N., Saruengkhanphasit, R., Eurtivong, C., Thasana, N., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 22
No.: 29
Page: 5924-5929
Published: 2024
doi: https://doi.org/10.1039/d4ob00630e

Molecular Reconstruction with Stereochemical Relay: An Investigation into the Rearrangement of Spiro[4.5]decadienone to Benzoxepane

By: Sittihan, S., Harada, S., Isono, T., Nemoto, T., and Ruchirawat, S.

Chemistry – An Asian Journal
Vol.: 19
No.: 2
Page:
Published: 2024
doi: https://doi.org/10.1002/asia.202300937

Novel naphthoquinones as potent aromatase inhibitors: Synthesis, anticancer, and in silico studies

By: Leechaisit, R., Mahalapbutr, P., Suriya, U., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., Prachayasittikul, V., and Pingaew, R.

Journal of Molecular Structure
Vol.: 1316
No.:
Page:
Published: 2024
doi: https://doi.org/10.1016/j.molstruc.2024.138981

Pharmacological Properties of White Mulberry (Morus alba L.) Leaves: Suppressing Migratory and Invasive Activities Against A549 Lung Cancer Cells

By: Srisomsap, C., Chaisuriya, P., Liana, D., Aiyarakanchanakun, P., Audsasan, T., Weeraphan, C., Svasti, J., and Phanumartwiwath, A.

Plant Foods for Human Nutrition
Vol.: 79
No.: 2
Page: 387-393
Published: 2024
doi: https://doi.org/10.1007/s11130-024-01184-9

Rapid and Scalable Production of Functional SARS-CoV-2 Virus-like Particles (VLPs) by a Stable HEK293 Cell Pool

By: Puarattana-aroonkorn, S., Tharakaraman, K., Suriyawipada, D., Ruchirawat, M., Fuangthong, M., Sasisekharan, R., and Artpradit, C.

Vaccines
Vol.: 12
No.: 6
Page:
Published: 2024
doi: https://doi.org/10.3390/vaccines12060561

A structure-based virtual high-throughput screening, molecular docking, molecular dynamics and MM/PBSA study identified novel putative drug-like dual inhibitors of trypanosomal cruzain and rhodesain cysteine proteases

By: Eurtivong, C., Zimmer, C., Schirmeister, T., Butkinaree, C., Saruengkhanphasit, R., Niwetmarin, W., Ruchirawat, S., and Bhambra, A. S.

Molecular Diversity
Vol.: 28
No.: 2
Page: 531-551
Published: 2024
doi: https://doi.org/10.1007/s11030-023-10600-2

Sultines as o -Quinodimethane Precursors in an Oxa-Diels-Alder Reaction: Synthesis of Functionalized Isochromans

By: Ngamnithiporn, A., Chuentragool, P., Songthammawat, P., Punnita, S., Photong, K., Ploypradith, P., and Ruchirawat, S.

Synlett
Vol.: 35
No.: 10
Page: 1180-1184
Published: 2024
doi: https://doi.org/10.1055/a-2236-9589

Synthesis, Antiacetylcholinesterase Activity, and Molecular Dynamics Simulation of Aporphine-benzylpyridinium Conjugates

By: Khunnawutmanotham, N., Sooknual, P., Batsomboon, P., Ploypradith, P., Chimnoi, N., Patigo, A., Saparpakorn, P., and Techasakul, S.

ACS Medicinal Chemistry Letters
Vol.: 15
No.: 1
Page: 132-142
Published: 2024
doi: https://doi.org/10.1021/acsmedchemlett.3c00467

Synthesis, in silico, in vitro evaluation of furanyl- and thiophenyl-3-phenyl-1H-indole-2-carbohydrazide derivatives as tubulin inhibitors and anticancer agents

By: Saruengkhanphasit, R., Ngiwsara, L., Lirdprapamongkol, K., Chatwichien, J., Niwetmarin, W., Eurtivong, C., Kittakoop, P., Svasti, J., and Ruchirawat, S.

RSC Medicinal Chemistry
Vol.: 15
No.: 7
Page: 2483-2495
Published: 2024
doi: https://doi.org/10.1039/d4md00210e

A toluidine blue/porous organic polymer/2D MoSe2 nanocomposite as an electrochemical signaling platform for a sensitive label-free aflatoxin B1 bioassay in some crops

By: Yaiwong, P., Iamsawat, K., Wiratchan, S., Jumpathong, W., Semakul, N., Bamrungsap, S., Jakmunee, J., and Ounnunkad, K.

Food Chemistry
Vol.: 439
No.:
Page:
Published: 2024
doi: https://doi.org/10.1016/j.foodchem.2023.138147

Two Cytochrome P450 Enzymes Form the Tricyclic Nested Skeleton of Meroterpenoids by Sequential Oxidative Reactions

By: Yang, E., Yao, Y., Su, H., Sun, Z., Gao, S. S., Sureram, S., Kittakoop, P., Fan, K., Pan, Y., Xu, X., Sun, Z. H., Ma, G., and Liu, G.

Journal of the American Chemical Society
Vol.:
No.:
Page:
Published: 2024
doi: https://doi.org/10.1021/jacs.4c01943

Two new serratene triterpenes from club moss cultivars

By: Thaisaeng, W., Thamnarak, W., Ruchirawat, S., Chainok, K., and Thasana, N.

Natural Product Research
Vol.: 38
No.: 15
Page: 2553-2561
Published: 2024
doi: https://doi.org/10.1080/14786419.2023.2188587

Unveiling Route for the Synthesis of Tröger’s Bases Through Azide Rearrangement

By: Jaithum, K., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.

Chemistry – An Asian Journal
Vol.: 19
No.: 17
Page:
Published: 2024
doi: https://doi.org/10.1002/asia.202400513

Vernonia amygdalina Leaf Extract Induces Apoptosis in HeLa Cells: A Metabolomics and Proteomics Study

By: Samutrtai, P., Yingchutrakul, Y., Faikhruea, K., Vilaivan, T., Chaikeeratisak, V., Chatwichien, J., Krobthong, S., and Aonbangkhen, C.

Pharmaceuticals
Vol.: 17
No.: 8
Page:
Published: 2024
doi: https://doi.org/10.3390/ph17081079

Visible Light-Induced One-Pot Carbonylation of Alkyl Halides with Aryl Formates

By: Chuentragool, P., Ngamnithiporn, A., Hongboon, P., and Ruchirawat, S.

Journal of Organic Chemistry
Vol.: 89
No.: 6
Page: 4205-4209
Published: 2024
doi: https://doi.org/10.1021/acs.joc.3c02763

2023

Altenusin inhibits epithelial to mesenchymal transition via suppression of TGF-β/MAPK signaling pathway in human renal proximal tubular cells and unilateral ureteral obstruction mice

By: Thipboonchoo, N., Sureram, S., Sa-nguansak, S., Kesornpun, C., Kittakoop, P., and Soodvilai, S.

Pharmaceutical Sciences Asia
Vol.: 50
No.: 4
Page: 371-380
Published: 2023
doi: https://doi.org/10.29090/psa.2023.04.23.645

The amide derivative of anticopalic acid induces non-apoptotic cell death in triple-negative breast cancer cells by inhibiting FAK activation

By: Chawengrum, P., Luepongpatthana, N., Thongnest, S., Sirirak, J., Boonsombat, J., Lirdprapamongkol, K., Keeratichamroen, S., Kongwaen, P., Montatip, P., Kittakoop, P., Svasti, J., and Ruchirawat, S.

Scientific Reports
Vol.: 13
No.: 1
Page:
Published: 2023
doi: https://doi.org/10.1038/s41598-023-40669-6

Aminochalcones Attenuate Neuronal Cell Death under Oxidative Damage via Sirtuin 1 Activity

By: Apiraksattayakul, S., Pingaew, R., Leechaisit, R., Prachayasittikul, V., Ruankham, W., Songtawee, N., Tantimongcolwat, T., Ruchirawat, S., Prachayasittikul, V., Prachayasittikul, S., and Phopin, K.

ACS Omega
Vol.: 8
No.: 37
Page: 33367-33379
Published: 2023
doi: https://doi.org/10.1021/acsomega.3c03047

Anthelmintic efficacy evaluation and mechanism of N-methylbenzo[d]oxazol-2-amine

By: Prangthip, P., Tummatorn, J., Adisakwattana, P., Uthailak, N., Boonyuen, U., Tipthara, P., Tarning, J., Laohapaisan, P., Thongsornkleeb, C., Ruchirawat, S., and Reamtong, O.

Scientific Reports
Vol.: 13
No.: 1
Page:
Published: 2023
doi: https://doi.org/10.1038/s41598-023-50305-y

Anti-Xanthine Oxidase 5′-Hydroxyhericenes A-D from the Edible Mushroom Hericium erinaceus and Structure Revision of 3-[2,3-Dihydroxy-4-(hydroxymethyl)tetrahydrofuran-1-yl]-pyridine-4,5-diol

By: Thongkongkaew, T., Jariyasopit, N., Khoomrung, S., Siritutsoontorn, S., Jitrapakdee, S., Kittakoop, P., and Ruchirawat, S.

ACS Omega
Vol.: 8
No.: 48
Page: 46284-46291
Published: 2023
doi: https://doi.org/10.1021/acsomega.3c07792

Base-Mediated and Silver-Catalyzed Divergent Synthesis of Hydroxynaphthalenamides and Phosphorylated Dihydronaphthylamides from Enone-Oxazolones

By: Worayuthakarn, R., Boontan, K., Chainok, K., Ruchirawat, S., and Thasana, N.

Journal of Organic Chemistry
Vol.: 88
No.: 23
Page: 16520-16538
Published: 2023
doi: https://doi.org/10.1021/acs.joc.3c01994

Bioisosteric Design Identifies Inhibitors of Mycobacterium tuberculosis DNA Gyrase ATPase Activity

By: Kamsri, B., Pakamwong, B., Thongdee, P., Phusi, N., Kamsri, P., Punkvang, A., Ketrat, S., Saparpakorn, P., Hannongbua, S., Sangswan, J., Suttisintong, K., Sureram, S., Kittakoop, P., Hongmanee, P., Santanirand, P., Leanpolchareanchai, J., Goudar, K. E., Spencer, J., Mulholland, A. J., and Pungpo, P.

Journal of Chemical Information and Modeling
Vol.: 63
No.: 9
Page: 2707-2718
Published: 2023
doi: https://doi.org/10.1021/acs.jcim.2c01376

Concise Synthesis of 1,4-Dideoxy-1,4-imino- l -arabinitol (LAB) from d -Xylose by Intramolecular Stereospecific Substitution of a Hydroxy Group

By: Akkarasamiyo, S., Na Sakonnakhon, H. P., Kuntiyong, P., Ploypradith, P., and Samec, J. S. M.

Synlett
Vol.: 34
No.: 5
Page: 441-444
Published: 2023
doi: https://doi.org/10.1055/s-0041-1738432

Copper-Catalyzed Guanylation by Ring Extension of 4-Hydroxyquinazoline for the Synthesis of Quinazolino[3,2-a]quinazolinones

By: Palavong, N., Arunkirirote, P., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.

Asian Journal of Organic Chemistry
Vol.: 12
No.: 6
Page:
Published: 2023
doi: https://doi.org/10.1002/ajoc.202300188

Cytotoxic Isopimarane Diterpenoids from Kaempferia koratensis Rhizomes

By: Kongwaen, P., Boonsombat, J., Thongnest, S., Ruchisansakun, S., Mahidol, C., and Ruchirawat, S.

Revista Brasileira de Farmacognosia
Vol.: 33
No.: 2
Page: 415-421
Published: 2023
doi: https://doi.org/10.1007/s43450-023-00359-w

Degradation of Methylene Blue Using Fly Ash as a Heterogeneous Fenton Catalyst

By: Saechan, C., Thawornpan, P., Thanapongpichat, S., Hongmanee, S., Srinoun, K., Win Tun, A., Tansila, N., Jumpathong, W., and Buncherd, H.

Analytical Letters
Vol.: 56
No.: 13
Page: 2099-2112
Published: 2023
doi: https://doi.org/10.1080/00032719.2022.2155179

Discovery of N-methylbenzo[d]oxazol-2-amine as new anthelmintic agent through scalable protocol for the synthesis of N-alkylbenzo[d]oxazol-2-amine and N-alkylbenzo[d]thiazol-2-amine derivatives

By: Laohapaisan, P., Reamtong, O., Tummatorn, J., Thongsornkleeb, C., Thaenkham, U., Adisakwattana, P., and Ruchirawat, S.

Bioorganic Chemistry
Vol.: 131
No.:
Page:
Published: 2023
doi: https://doi.org/10.1016/j.bioorg.2022.106287

Discovery of Novel Naphthoquinone-Chalcone Hybrids as Potent FGFR1 Tyrosine Kinase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling

By: Leechaisit, R., Mahalapbutr, P., Boonsri, P., Karnchanapandh, K., Rungrotmongkol, T., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., Prachayasittikul, V., and Pingaew, R.

ACS Omega
Vol.: 8
No.: 36
Page: 32593-32605
Published: 2023
doi: https://doi.org/10.1021/acsomega.3c03176

Divergent synthesis of 3,4-dihydro-2H-benzo[h]chromen-2-one and fluorenone derivatives from ortho-alkynylarylketones

By: Jantrapirom, J., Palavong, N., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 21
No.: 44
Page: 8888-8901
Published: 2023
doi: https://doi.org/10.1039/d3ob01492d

Divergent Synthesis of Isochroman-4-ols, 1,3-Dihydroisobenzofurans, and Tetrahydro-2 H -indeno[2,1- b ]furan-2-ones via Epoxidation/Cyclization Strategy of (E)-(2-Stilbenyl/Styrenyl)methanols

By: Jongcharoenkamol, J., Jancharoen, K., Batsomboon, P., Ruchirawat, S., and Ploypradith, P.

Synthesis (Germany)
Vol.: 55
No.: 17
Page: 2757-2772
Published: 2023
doi: https://doi.org/10.1055/s-0042-1751458

Fabrication, Optimization, and Characterization of Antibacterial Electrospun Shellac Fibers Loaded with Kaempferia parviflora Extract

By: Krongrawa, W., Limmatvapirat, S., Vollrath, M. K., Kittakoop, P., Saibua, S., and Limmatvapirat, C.

Pharmaceutics
Vol.: 15
No.: 1
Page:
Published: 2023
doi: https://doi.org/10.3390/pharmaceutics15010123

Halogenative Annulation Reactions of Alkyne-Tethered N – And O -Containing Arenes: Methods for Accessing Aryl-Fused Halogenated N – And O -Heterocycles

By: Tummatorn, J., Ruchirawat, S., and Thongsornkleeb, C.

Synthesis (Germany)
Vol.: 55
No.: 19
Page: 3073-3089
Published: 2023
doi: https://doi.org/10.1055/a-2114-7582

In vitro evaluation of the anti-breast cancer properties and gene expression profiles of Thai traditional formulary medicine extracts

By: Khamwut, A., Klomkliew, P., Jumpathong, W., Kaewsapsak, P., Chanchaem, P., Sivapornnukul, P., Chantanakat, K., T-Thienprasert, N. P., and Payungporn, S.

Biomedical Reports
Vol.: 19
No.: 4
Page:
Published: 2023
doi: https://doi.org/10.3892/br.2023.1652

Kaemtakols A–D, highly oxidized pimarane diterpenoids with potent anti-inflammatory activity from Kaempferia takensis

By: Jongsomjainuk, O., Boonsombat, J., Thongnest, S., Prawat, H., Batsomboon, P., Charoensutthivarakul, S., Ruchisansakun, S., Chainok, K., Sirirak, J., Mahidol, C., and Ruchirawat, S.

Natural Products and Bioprospecting
Vol.: 13
No.: 1
Page:
Published: 2023
doi: https://doi.org/10.1007/s13659-023-00420-0

A Mechanistically Deceiving Formation of Aryl(1-indanyl)ketones via Acid-Catalyzed Cyclization of ortho-Alkynylarylmethanols

By: Rodphon, W., Linkhum, S., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.

Journal of Organic Chemistry
Vol.: 88
No.: 7
Page: 4172-4186
Published: 2023
doi: https://doi.org/10.1021/acs.joc.2c02664

Microwave-assisted commercial copper-catalyzed aerobic oxidative synthesis of AChE quinazolinone inhibitors under solvent free conditions

By: Jongcharoenkamol, J., Naksing, P., Nimnuan, N., Singh, T., Chatwichien, J., Temkitthawon, P., Sriwattanawarunyoo, C., Choommongkol, V., Meepowpan, P., and Kerdphon, S.

RSC Advances
Vol.: 13
No.: 39
Page: 27657-27662
Published: 2023
doi: https://doi.org/10.1039/d3ra05739a

Mn(OAc)3-Mediated One-Pot Condensation-Oxidative Annulation of 2-Alkynylanilines and 1,3-Ketoesters: Synthesis of 2-Substituted Quinolines

By: Punjajom, K., Ruengsangtongkul, S., Tummatorn, J., Paiboonsombat, P., Ruchirawat, S., and Thongsornkleeb, C.

Journal of Organic Chemistry
Vol.: 88
No.: 11
Page: 6736-6749
Published: 2023
doi: https://doi.org/10.1021/acs.joc.3c00027

Novel Pd(ii) pincer complexes bearing salicylaldimine-based benzothiazole derivatives: synthesis, structural characterization, DNA/BSA binding, and biological evaluation

By: Wongsuwan, S., Chatwichien, J., Sirisaksoontorn, W., Chainok, K., Songsasen, A., and Chotima, R.

New Journal of Chemistry
Vol.: 47
No.: 22
Page: 10624-10637
Published: 2023
doi: https://doi.org/10.1039/d3nj00458a

Phlegcarines A-C, three Lycopodium alkaloids from Phlegmariurus carinatus (Desv. ex Poir.) Ching

By: Thamnarak, W., Thaisaeng, W., Batsomboon, P., Eurtivong, C., Wannarit, N., Ruchirawat, S., and Thasana, N.

Phytochemistry
Vol.: 206
No.:
Page:
Published: 2023
doi: https://doi.org/10.1016/j.phytochem.2022.113553

Phukettosides A–E, mono- and bis-iridoid glycosides, from the leaves of Morinda umbellata L

By: Kaweetripob, W., Thongnest, S., Boonsombat, J., Batsomboon, P., Salae, A. W., Prawat, H., Mahidol, C., and Ruchirawat, S.

Phytochemistry
Vol.: 216
No.:
Page:
Published: 2023
doi: https://doi.org/10.1016/j.phytochem.2023.113890

Protein Modification via Nitrile Oxide−Dehydroalanine Cycloaddition: Formation of Isoxazoline Ring on the Protein Backbone

By: Phanumartwiwath, A., Kesornpun, C., Chokchaichamnankit, D., Khongmanee, A., Diskul-Na-Ayudthaya, P., Ruangjaroon, T., Srisomsap, C., Kittakoop, P., Svasti, J., and Ruchirawat, S.

ChemBioChem
Vol.: 24
No.: 20
Page:
Published: 2023
doi: https://doi.org/10.1002/cbic.202300268

Rapid synthesis of α(1,2)-D-mannans on the surface of Mycobacterium tuberculosis and their nitric oxide-inducing activities

By: Suwanwong, N., Chatwichien, J., Ruchirawat, S., and Boonyarattanakalin, S.

Carbohydrate Polymer Technologies and Applications
Vol.: 6
No.:
Page:
Published: 2023
doi: https://doi.org/10.1016/j.carpta.2023.100375

The redox-sensing mechanism of Agrobacterium tumefaciens NieR as a thiol-based oxidation sensor for hypochlorite stress

By: Nontaleerak, B., Eurtivong, C., Weeraphan, C., Buncherd, H., Chokchaichamnankit, D., Srisomsap, C., Svasti, J., Sukchawalit, R., and Mongkolsuk, S.

Free Radical Biology and Medicine
Vol.: 208
No.:
Page: 211-220
Published: 2023
doi: https://doi.org/10.1016/j.freeradbiomed.2023.08.002

Schomburginones A‒J, geranylated benzophenones from the leaves of Garcinia schomburgkiana and their cytotoxic and anti-inflammatory activities

By: Sukandar, E. R., Kaennakam, S., Wongsuwan, S., Chatwichien, J., Krobthong, S., Yingchutrakul, Y., Mahatnirunkul, T., Mulya, F., Parasuk, V., Harding, D. J., Poldorn, P., Rungrotmongkol, T., Tip-pyang, S., Aonbangkhen, C., and Chavasiri, W.

Phytochemistry
Vol.: 211
No.:
Page:
Published: 2023
doi: https://doi.org/10.1016/j.phytochem.2023.113701

Selective electrophilic cyclization of ortho-carbonylarylacetylenols for the synthesis of cyclopenta[a]naphthalenol and 2-phenylnaphthalen-1-ol analogs

By: Jantrapirom, J., Yongpanich, P., Tummatorn, J., Chainok, K., Jiajaroen, S., Thongsornkleeb, C., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 21
No.: 42
Page: 8500-8515
Published: 2023
doi: https://doi.org/10.1039/d3ob01344h

Synthesis of Clausena Alkaloids Using Unique Ring Expansion of Dihydroisoquinolines and Their Cholinesterase Inhibitory Activity

By: Worayuthakarn, R., Ngernnak, C., Ruchirawat, S., Chainok, K., Wannarit, N., and Thasana, N.

Synthesis (Germany)
Vol.: 55
No.: 14
Page: 2241-2252
Published: 2023
doi: https://doi.org/10.1055/s-0042-1752658

Synthesis of Naphtho[2,3-d]oxazoles via Ag(I) Acid-Mediated Oxazole-Benzannulation of ortho-Alkynylamidoarylketones

By: Rodphon, W., Jaithum, K., Linkhum, S., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.

Journal of Organic Chemistry
Vol.: 88
No.: 5
Page: 2677-2691
Published: 2023
doi: https://doi.org/10.1021/acs.joc.2c00940

Three-Component Aza-Diels-Alder Reaction for the Syntheses of Tetrahydroisoquinoline Derivatives

By: Ngamnithiporn, A., Chuentragool, P., Ploypradith, P., and Ruchirawat, S.

Asian Journal of Organic Chemistry
Vol.: 12
No.: 9
Page:
Published: 2023
doi: https://doi.org/10.1002/ajoc.202300366

UHPLC-QQQ-MS and RP-HPLC Detection of Bioactive Alizarin and Scopoletin Metabolites from Morinda citrifolia Root Extracts and Their Antitubercular, Antibacterial, and Antioxidant Activities

By: Sam-Ang, P., Phanumartwiwath, A., Liana, D., Sureram, S., Hongmanee, P., and Kittakoop, P.

ACS Omega
Vol.: 8
No.: 32
Page: 29615-29624
Published: 2023
doi: https://doi.org/10.1021/acsomega.3c03656

Virucidal and Antiviral Polyhydroxylated Fatty Alcohols in Avocado Fruit Pulp (Persea americana) of Booth 7 Cultivar¶

By: Darshana, D., Chutiwitoonchai, N., Paemanee, A., Sureram, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.

ACS Food Science and Technology
Vol.: 3
No.: 10
Page: 1759-1767
Published: 2023
doi: https://doi.org/10.1021/acsfoodscitech.3c00326

2022

4b-Aryltetrahydroindeno[1,2- a ]indenes by Acid-Catalyzed Transannular Cyclization of Benzannulated Cyclooctene Alcohols

By: Songthammawat, P., Phumjan, T., Ruchirawat, S., and Ploypradith, P.

Synlett
Vol.: 33
No.: 14
Page: 1312-1316
Published: 2022
doi: https://doi.org/10.1055/a-1778-8143

Acetogenins from the stems of Uvaria micrantha showing antiproliferative effects on HepG2 liver cancer cells

By: Thongnest, S., Boonsombat, J., Keeratichamroen, S., Lirdprapamongkol, K., Kaweetripob, W., Kheawchaum, S., Mahidol, C., Svasti, J., Ruchirawat, S., and Prawat, H.

Phytochemistry
Vol.: 204
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.phytochem.2022.113450

Acid-dependent Divergent Conversion of ortho-Arylcyclopropanecarbonyl Carboxaldehydes for the Synthesis of Furanodibenzocycloheptenes and Dibenzocycloheptenes

By: Palavong, N., Jantrapirom, J., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.

Asian Journal of Organic Chemistry
Vol.: 11
No.: 10
Page:
Published: 2022
doi: https://doi.org/10.1002/ajoc.202200507

Ag(I)-Catalyzed/Acid-Mediated Cascade Cyclization of ortho-Alkynylaryl-1,3-dicarbonyls to Access Arylnaphthalenelactones and Furanonaphthol Libraries via Aryl-Disengagement

By: Laohapaisan, P., Lumyong, K., Tummatorn, J., Thongsornkleeb, C., Chatwichien, J., Supantanapong, N., and Ruchirawat, S.

Chemistry – An Asian Journal
Vol.: 17
No.: 1
Page:
Published: 2022
doi: https://doi.org/10.1002/asia.202101212

ALKALOIDS AND ALKALOID-LIKE COMPOUNDS ARE POTENTIAL SCAFFOLDS OF ANTIVIRAL AGENTS AGAINST SARS-COV-2 (COVID-19) VIRUS

By: Kittakoop, P., Darshana, D., Sangsuwan, R., and Mahidol, C.

Heterocycles
Vol.: 105
No.: 1
Page: 115-146
Published: 2022
doi: https://doi.org/10.3987/REV-22-SR(R)3

Anticancer activity and QSAR study of sulfur-containing thiourea and sulfonamide derivatives

By: Pingaew, R., Prachayasittikul, V., Worachartcheewan, A., Thongnum, A., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.

Heliyon
Vol.: 8
No.: 8
Page:
Published: 2022
doi: https://doi.org/10.1016/j.heliyon.2022.e10067

Asymmetric Total Synthesis and Structure Elucidation of Huperzine H

By: Shiomi, S., Wilailak, K., Soutome, W., Takayama, H., Kitajima, M., and Ishikawa, H.

Journal of Organic Chemistry
Vol.: 87
No.: 5
Page: 3730-3735
Published: 2022
doi: https://doi.org/10.1021/acs.joc.1c02672

Biosurfactant-Producing Bacillus velezensis PW192 as an Anti-Fungal Biocontrol Agent against Colletotrichum gloeosporioides and Colletotrichum musae

By: Jumpathong, W., Intra, B., Euanorasetr, J., and Wanapaisan, P.

Microorganisms
Vol.: 10
No.: 5
Page:
Published: 2022
doi: https://doi.org/10.3390/microorganisms10051017

Ceric Ammonium Nitrate Promoted Oxidative Coupling of Terminal Alkynes and 1,3-Keto Esters: A Synthesis of Unsymmetrical 1,1,2-Triacylalkenes

By: Ruengsangtongkul, S., Kuribara, T., Chaisan, N., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.

Synlett
Vol.: 33
No.: 14
Page: 1329-1334
Published: 2022
doi: https://doi.org/10.1055/a-1774-6966

Characterisation of the triclosan efflux pump TriABC and its regulator TriR in Agrobacterium tumefaciens C58

By: Nontaleerak, B., Tasnawijitwong, N., Eurtivong, C., Sirikanchana, K., Satayavivad, J., Sukchawalit, R., and Mongkolsuk, S.

Microbiological Research
Vol.: 263
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.micres.2022.127112

A Compilation of Synthetic Strategies to Access the Most Utilized Indoloquinoline Motifs

By: Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.

Chemistry – An Asian Journal
Vol.: 17
No.: 7
Page:
Published: 2022
doi: https://doi.org/10.1002/asia.202200040

Copper-Mediated C-O/C-N Bond Formation: A Facile Synthesis of 3-Amidocoumarin, 3-Amidoazacoumarin, and N -Aroylindole Derivatives

By: Worayuthakarn, R., Suddee, N., Nealmongkol, P., Ruchirawat, S., and Thasana, N.

Synlett
Vol.: 33
No.: 14
Page: 1431-1437
Published: 2022
doi: https://doi.org/10.1055/a-1784-1973

Cytotoxic isoflavonoids from the roots of Desmodium velutinum (Willd.) DC

By: Kaweetripob, W., Thongnest, S., Boonsombat, J., Kheawchaum, S., Mahidol, C., Prawat, H., and Ruchirawat, S.

Phytochemistry Letters
Vol.: 48
No.:
Page: 47-53
Published: 2022
doi: https://doi.org/10.1016/j.phytol.2022.01.018

The Design and Synthesis of a New Series of 1,2,3-Triazole-Cored Structures Tethering Aryl Urea and Their Highly Selective Cytotoxicity toward HepG2

By: Oekchuae, S., Sirirak, J., Charoensuksai, P., Wongprayoon, P., Chuaypen, N., Boonsombat, J., Ruchirawat, S., Tangkijvanich, P., Suksamrarn, A., and Limpachayaporn, P.

Pharmaceuticals
Vol.: 15
No.: 5
Page:
Published: 2022
doi: https://doi.org/10.3390/ph15050504

Dihalooxygenation of Alkynes and Alkynols: Preparation of 2,2-Dihaloketones and gem -Dihalolactols

By: Chaisan, N., Ruengsangtongkul, S., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.

Synlett
Vol.: 33
No.: 14
Page: 1426-1430
Published: 2022
doi: https://doi.org/10.1055/a-1774-7077

Discovery of Anilino-1,4-naphthoquinones as Potent EGFR Tyrosine Kinase Inhibitors: Synthesis, Biological Evaluation, and Comprehensive Molecular Modeling

By: Mahalapbutr, P., Leechaisit, R., Thongnum, A., Todsaporn, D., Prachayasittikul, V., Rungrotmongkol, T., Prachayasittikul, S., Ruchirawat, S., Prachayasittikul, V., and Pingaew, R.

ACS Omega
Vol.: 7
No.: 21
Page: 17881-17893
Published: 2022
doi: https://doi.org/10.1021/acsomega.2c01188

Discovery of nitric oxide-inducing activities of synthetic LAM glycan motifs prepared by scalable rapid syntheses

By: Suwanwong, N., Chatwichien, J., Chainok, K., Ruchirawat, S., and Boonyarattanakalin, S.

Carbohydrate Polymers
Vol.: 296
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.carbpol.2022.119637

Discovery of novel and potent InhA inhibitors by an in silico screening and pharmacokinetic prediction

By: Hanwarinroj, C., Phusi, N., Kamsri, B., Kamsri, P., Punkvang, A., Ketrat, S., Saparpakorn, P., Hannongbua, S., Suttisintong, K., Kittakoop, P., Spencer, J., Mulholland, A. J., and Pungpo, P.

Future Medicinal Chemistry
Vol.: 14
No.: 10
Page: 717-729
Published: 2022
doi: https://doi.org/10.4155/fmc-2021-0348

Discovery of potent antiproliferative agents from selected oxygen heterocycles as EGFR tyrosine kinase inhibitors from the U.S. National Cancer Institute database by in silico screening and bioactivity evaluation

By: Jiwacharoenchai, N., Saruengkhanphasit, R., Niwetmarin, W., Seetaha, S., Choowongkomon, K., Ruchirawat, S., and Eurtivong, C.

Bioorganic and Medicinal Chemistry Letters
Vol.: 58
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.bmcl.2021.128524

Diterpenoids and p-methoxycinnamic acid diol esters from Kaempferia saraburiensis Picheans. (Zingiberaceae): Structural assignment of saraburol and their biological activities

By: Booranaseensuntorn, P., Boonsombat, J., Mahidol, C., Reuk-Ngam, N., Khlaychan, P., Batsomboon, P., Techasakul, S., Thongnest, S., and Ruchirawat, S.

Phytochemistry
Vol.: 199
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.phytochem.2022.113181

Dulcisenes C-E, polyoxygenated cyclohexenes, from Uvaria dulcis dunal and their cytotoxic activity

By: Pailee, P., Ploypradith, P., Mahidol, C., Ruchirawat, S., and Prachyawarakorn, V.

Phytochemistry
Vol.: 202
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.phytochem.2022.113298

Ent-abietane diterpenoid lactone glycosides and a phenolic glycoside from Phlogacanthus pulcherrimus T. Anderson with cytotoxic and cancer chemopreventive activities

By: Kheawchaum, S., Mahidol, C., Thongnest, S., Boonsombat, J., Batsomboon, P., Sitthimonchai, S., Ruchirawat, S., and Prawat, H.

Phytochemistry
Vol.: 201
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.phytochem.2022.113261

Facile synthesis of 1-substituted 4-H phthalazine, a versatile scaffold for chemically diverse phthalazines

By: Hadsarung, R., Thongnest, S., Oekchuae, S., Chaiyaveij, D., Boonsombat, J., and Ruchirawat, S.

Tetrahedron
Vol.: 121
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.tet.2022.132920

Functionalized Chromans from ortho-Quinone Methides and Arylallenes

By: Akkarasereenon, K., Batsomboon, P., Ruchirawat, S., and Ploypradith, P.

Journal of Organic Chemistry
Vol.: 87
No.: 23
Page: 15863-15887
Published: 2022
doi: https://doi.org/10.1021/acs.joc.2c01962

Hybrid Plasticizers Enhance Specificity and Sensitivity of an Electrochemical-Based Sensor for Cadmium Detection

By: Ruangsuj, P., Wanthongcharoen, S., Chaisriratanakul, W., Bunjongpru, W., Yamprayoonswat, W., Jeamsaksiri, W., Jumpathong, W., and Yasawong, M.

International Journal of Molecular Sciences
Vol.: 23
No.: 12
Page:
Published: 2022
doi: https://doi.org/10.3390/ijms23126402

Identification of Potent DNA Gyrase Inhibitors Active against Mycobacterium tuberculosis

By: Pakamwong, B., Thongdee, P., Kamsri, B., Phusi, N., Kamsri, P., Punkvang, A., Ketrat, S., Saparpakorn, P., Hannongbua, S., Ariyachaokun, K., Suttisintong, K., Sureram, S., Kittakoop, P., Hongmanee, P., Santanirand, P., Spencer, J., Mulholland, A. J., and Pungpo, P.

Journal of Chemical Information and Modeling
Vol.: 62
No.: 7
Page: 1680-1690
Published: 2022
doi: https://doi.org/10.1021/acs.jcim.1c01390

Impact of the ferrocenyl group on cytotoxicity and KSP inhibitory activity of ferrocenyl monastrol conjugates

By: Wieczorek-Błauż, A., Kowalczyk, K., Błauż, A., Makal, A., Pawlȩdzio, S., Eurtivong, C., Arabshahi, H. J., Reynisson, J., Hartinger, C. G., Rychlik, B., and Plażuk, D.

Dalton Transactions
Vol.: 51
No.: 2
Page: 491-508
Published: 2022
doi: https://doi.org/10.1039/d1dt03553c

In silico design of novel quinazoline-based compounds as potential Mycobacterium tuberculosis PknB inhibitors through 2D and 3D-QSAR, molecular dynamics simulations combined with pharmacokinetic predictions

By: Hanwarinroj, C., Thongdee, P., Sukchit, D., Taveepanich, S., Kamsri, P., Punkvang, A., Ketrat, S., Saparpakorn, P., Hannongbua, S., Suttisintong, K., Kittakoop, P., Spencer, J., Mulholland, A. J., and Pungpo, P.

Journal of Molecular Graphics and Modelling
Vol.: 115
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.jmgm.2022.108231

Inhibition of Mycobacterium tuberculosis InhA by 3-nitropropanoic acid

By: Songsiriritthigul, C., Hanwarinroj, C., Pakamwong, B., Srimanote, P., Suttipanta, N., Sureram, S., Suttisintong, K., Kamsri, P., Punkvang, A., Spencer, J., Kittakoop, P., and Pungpo, P.

Proteins: Structure, Function and Bioinformatics
Vol.: 90
No.: 3
Page: 898-904
Published: 2022
doi: https://doi.org/10.1002/prot.26268

JAK2/STAT3-mediated dose-dependent cytostatic and cytotoxic effects of sesquiterpene lactones from Gymnanthemum extensum on A549 human lung carcinoma cells

By: Keeratichamroen, S., Lirdprapamongkol, K., Thongnest, S., Boonsombat, J., Chawengrum, P., Sornprachum, T., Sirirak, J., Verathamjamras, C., Ornnork, N., Ruchirawat, S., and Svasti, J.

Oncology Reports
Vol.: 47
No.: 1
Page:
Published: 2022
doi: https://doi.org/10.3892/or.2021.8217

LC-MS/MS metabolomics-facilitated identification of the active compounds responsible for anti-allergic activity of the ethanol extract of Xenostegia tridentata

By: Suntivich, R., Songjang, W., Jiraviriyakul, A., Ruchirawat, S., and Chatwichien, J.

PloS One
Vol.: 17
No.: 4 April
Page:
Published: 2022
doi: https://doi.org/10.1371/journal.pone.0265505

Lipase-catalyzed esterification in water enabled by nanomicelles. Applications to 1-pot multi-step sequences

By: Singhania, V., Cortes-Clerget, M., Dussart-Gautheret, J., Akkachairin, B., Yu, J., Akporji, N., Gallou, F., and Lipshutz, B. H.

Chemical Science
Vol.: 13
No.: 5
Page: 1440-1445
Published: 2022
doi: https://doi.org/10.1039/d1sc05660c

Novel psoralen derivatives as anti-breast cancer agents and their light-activated cytotoxicity against HER2 positive breast cancer cells

By: Aekrungrueangkit, C., Wangngae, S., Kamkaew, A., Ardkhean, R., Thongnest, S., Boonsombat, J., Ruchirawat, S., and Khotavivattana, T.

Scientific Reports
Vol.: 12
No.: 1
Page:
Published: 2022
doi: https://doi.org/10.1038/s41598-022-17625-x

OXIDATIVE FRAGMENTATION OF CYTISINE AS AN ENTRY TO THE BIS(PIPERIDINE) SCAFFOLD OF VIRGIDIVARINE

By: Niwetmarin, W., and Gallagher, T.

Heterocycles
Vol.: 105
No.: 1
Page: 500-510
Published: 2022
doi: https://doi.org/10.3987/COM-22-S(R)21

The Peptide A-3302-B Isolated from a Marine Bacterium Micromonospora sp. Inhibits HSV-2 Infection by Preventing the Viral Egress from Host Cells

By: Sureram, S., Arduino, I., Ueoka, R., Rittà, M., Francese, R., Srivibool, R., Darshana, D., Piel, J., Ruchirawat, S., Muratori, L., Lembo, D., Kittakoop, P., and Donalisio, M.

International Journal of Molecular Sciences
Vol.: 23
No.: 2
Page:
Published: 2022
doi: https://doi.org/10.3390/ijms23020947

Photoinduced C-C bond cleavage for the synthesis of 2,4-disubstituted-1-naphthols from indenone derivatives and sulfoxonium ylide

By: Khorphueng, P., Tummatorn, J., Patumanon, W., Thongsornkleeb, C., Chonradeenitchakul, S., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 20
No.: 28
Page: 5520-5524
Published: 2022
doi: https://doi.org/10.1039/d2ob00958g

Siamenflavones A-C, three undescribed biflavonoids from Selaginella siamensis Hieron. and biflavonoids from spike mosses as EGFR inhibitor

By: Demehin, A. A., Thamnarak, W., Lamtha, T., Chatwichien, J., Eurtivong, C., Choowongkomon, K., Chainok, K., Ruchirawat, S., and Thasana, N.

Phytochemistry
Vol.: 203
No.:
Page:
Published: 2022
doi: https://doi.org/10.1016/j.phytochem.2022.113374

Synergistic Lewis-Brønsted Acid Catalysis in Cascade Cyclization of ortho-Alkynylaryl Cyclopropylketones for the Synthesis of 2,3-Dihydronaphtho[1,2- b]furans

By: Jaithum, K., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.

Journal of Organic Chemistry
Vol.: 87
No.: 22
Page: 15358-15379
Published: 2022
doi: https://doi.org/10.1021/acs.joc.2c01940

Syntheses of 3-Aryl Tetrahydroisoquinolines via an Intermolecular [4 + 2] Cycloaddition of Sultines with Imines

By: Ngamnithiporn, A., Chuentragool, P., Ploypradith, P., and Ruchirawat, S.

Organic Letters
Vol.: 24
No.: 23
Page: 4192-4196
Published: 2022
doi: https://doi.org/10.1021/acs.orglett.2c01437

Synthesis and Anticancer Activity of Pentafluorobenzenesulfonamide Derivatives as Caspase-Dependent Apoptosis-Inducing Agents

By: Sittihan, S., Sopha, P., and Ruchirawat, S.

ChemMedChem
Vol.: 17
No.: 3
Page:
Published: 2022
doi: https://doi.org/10.1002/cmdc.202100637

SYNTHESIS OF ACETAMIDOSULFONAMIDE DERIVATIVES WITH ANTIOXIDATIVE AND QSAR STUDIES

By: Worachartcheewan, A., Pisutjaroenpong, S., Pingaew, R., Prachayasittikul, S., Siriwong, S., Ruchirawat, S., and Prachayasittikul, V.

EXCLI journal
Vol.: 21
No.:
Page: 360-379
Published: 2022
doi: https://doi.org/10.17179/excli2021-4590

Synthesis of Chiral Tetrahydro-3-benzazepine Motifs by Iridium-Catalyzed Asymmetric Hydrogenation of Cyclic Ene-carbamates

By: Peters, B. B. C., Andersson, P. G., Ruchirawat, S., and Ieawsuwan, W.

Organic Letters
Vol.: 24
No.: 10
Page: 1969-1973
Published: 2022
doi: https://doi.org/10.1021/acs.orglett.2c00362

SYNTHESIS OF NOVEL FLUORESCENT BICYCLIC AMIDINES AND EVALUATION OF THEIR PHOTOPHYSICAL PROPERTIES

By: Disadee, W., Trisupphakant, K., and Ruchirawat, S.

Heterocycles
Vol.: 105
No.: 1
Page: 417-437
Published: 2022
doi: https://doi.org/10.3987/COM-22-S(R)13

Total Synthesis of Palodesangrens A and C

By: Tangdenpaisal, K., Songthammawat, P., Ruchirawat, S., and Ploypradith, P.

Journal of Organic Chemistry
Vol.: 87
No.: 1
Page: 386-398
Published: 2022
doi: https://doi.org/10.1021/acs.joc.1c02417

Total Synthesis of Pentaketide Ansamycin Microansamycin H

By: Sittihan, S., and Ruchirawat, S.

Organic Letters
Vol.: 24
No.: 24
Page: 4470-4473
Published: 2022
doi: https://doi.org/10.1021/acs.orglett.2c01760

Traveling Wave Ion Mobility-Derived Collision Cross Section Database for Plant Specialized Metabolites: An Application to Ventilago harmandiana Pierre

By: Jariyasopit, N., Limjiasahapong, S., Kurilung, A., Sartyoungkul, S., Wisanpitayakorn, P., Nuntasaen, N., Kuhakarn, C., Reutrakul, V., Kittakoop, P., Sirivatanauksorn, Y., and Khoomrung, S.

Journal of Proteome Research
Vol.: 21
No.: 10
Page: 2481-2492
Published: 2022
doi: https://doi.org/10.1021/acs.jproteome.2c00413

Two new nor-lignans, siamensinols A and B, from Selaginella siamensis Hieron. and their biological activities

By: Thamnarak, W., Eurtivong, C., Pollawatn, R., Ruchirawat, S., and Thasana, N.

Natural Product Research
Vol.: 36
No.: 21
Page: 5591-5599
Published: 2022
doi: https://doi.org/10.1080/14786419.2021.2022664

Virtual Screening Identifies Novel and Potent Inhibitors of Mycobacterium tuberculosis PknB with Antibacterial Activity

By: Thongdee, P., Hanwarinroj, C., Pakamwong, B., Kamsri, P., Punkvang, A., Leanpolchareanchai, J., Ketrat, S., Saparpakorn, P., Hannongbua, S., Ariyachaokun, K., Suttisintong, K., Sureram, S., Kittakoop, P., Hongmanee, P., Santanirand, P., Mukamolova, G. V., Blood, R. A., Takebayashi, Y., Spencer, J., Mulholland, A. J., and Pungpo, P.

Journal of Chemical Information and Modeling
Vol.: 62
No.: 24
Page: 6508-6518
Published: 2022
doi: https://doi.org/10.1021/acs.jcim.2c00531

Virucidal Activity of Essential Oils From Citrus x aurantium L. Against Influenza A Virus H1N1: Limonene as a Potential Household Disinfectant Against Virus

By: Fadilah, N. Q., Jittmittraphap, A., Leaungwutiwong, P., Pripdeevech, P., Dhanushka, D., Mahidol, C., Ruchirawat, S., and Kittakoop, P.

Natural Product Communications
Vol.: 17
No.: 1
Page:
Published: 2022
doi: https://doi.org/10.1177/1934578X211072713

2021

The 4-(Phenylsulfanyl) butan-2-one Improves Impaired Fear Memory Retrieval and Reduces Excessive Inflammatory Response in Triple Transgenic Alzheimer’s Disease Mice

By: Varinthra, P., Ganesan, K., Huang, S. P., Chompoopong, S., Eurtivong, C., Suresh, P., Wen, Z. H., and Liu, I. Y.

Frontiers in Aging Neuroscience
Vol.: 13
No.:
Page:
Published: 2021
doi: https://doi.org/10.3389/fnagi.2021.615079

Antitubercular and antibacterial activities of isoxazolines derived from natural products: Isoxazolines as inhibitors of Mycobacterium tuberculosis InhA

By: Phanumartwiwath, A., Kesornpun, C., Sureram, S., Hongmanee, P., Pungpo, P., Kamsri, P., Punkvang, A., Eurtivong, C., Kittakoop, P., and Ruchirawat, S.

Journal of Chemical Research
Vol.: 45
No.: 11-12
Page: 1003-1015
Published: 2021
doi: https://doi.org/10.1177/17475198211047801

Chemoenzymatic and Protecting-Group-Free Synthesis of 1,4-Substituted 1,2,3-Triazole-α- d -glucosides with Potent Inhibitory Activity toward Lysosomal α-Glucosidase

By: Gorantla, J. N., Maniganda, S., Pengthaisong, S., Ngiwsara, L., Sawangareetrakul, P., Chokchaisiri, S., Kittakoop, P., Svasti, J., and Ketudat Cairns, J. R.

ACS Omega
Vol.: 6
No.: 39
Page: 25710-25719
Published: 2021
doi: https://doi.org/10.1021/acsomega.1c03928

Dibrominative Spirocyclization of 2-Butynolyl Anilides: Synthesis of gem-Dibromospirocyclic Benzo[ d][1,3]oxazines and Their Application in the Synthesis of 4 H-Furo[3,2- b]indoles

By: Chaisan, N., Ruengsangtongkul, S., Tummatorn, J., Ruchirawat, S., Chainok, K., and Thongsornkleeb, C.

Journal of Organic Chemistry
Vol.: 86
No.: 6
Page: 4671-4698
Published: 2021
doi: https://doi.org/10.1021/acs.joc.1c00086

The discovery of novel antitrypanosomal 4-phenyl-6-(pyridin-3-yl)pyrimidines

By: Robinson, W. J., Taylor, A. E., Lauga-Cami, S., Weaver, G. W., Arroo, R. R. J., Kaiser, M., Gul, S., Kuzikov, M., Ellinger, B., Singh, K., Schirmeister, T., Botana, A., Eurtivong, C., and Bhambra, A. S.

European Journal of Medicinal Chemistry
Vol.: 209
No.:
Page:
Published: 2021
doi: https://doi.org/10.1016/j.ejmech.2020.112871

Diterpenoids with Aromatase Inhibitory Activity from the Rhizomes of Kaempferia elegans

By: Chawengrum, P., Boonsombat, J., Mahidol, C., Eurtivong, C., Kittakoop, P., Thongnest, S., and Ruchirawat, S.

Journal of Natural Products
Vol.: 84
No.: 6
Page: 1738-1747
Published: 2021
doi: https://doi.org/10.1021/acs.jnatprod.0c01292

An Expeditious Modular Hybrid Strategy for the Diversity-Oriented Synthesis of Lamellarins/Azalamellarins with Anticancer Cytotoxicity

By: Klumthong, K., Chalermsub, P., Sopha, P., Ruchirawat, S., and Ploypradith, P.

Journal of Organic Chemistry
Vol.: 86
No.: 21
Page: 14883-14902
Published: 2021
doi: https://doi.org/10.1021/acs.joc.1c01639

Genome sequence of streptomyces cavourensis BUU135, isolated from soil from a tropical fruit farm in Thailand

By: Tangwattanachuleeporn, M., Ruangsuj, P., Yamprayoonswat, W., Sittihan, S., Jumpathong, W., and Yasawong, M.

Microbiology resource announcements
Vol.: 10
No.: 19
Page:
Published: 2021
doi: https://doi.org/10.1128/MRA.01428-20

Highly Regioselective Tandem Reaction of Ene-Yne-Oxazolones Induced by H-Phosphonates: Construction of Phosphinylindane Derivatives

By: Worayuthakarn, R., Deesiri, S., Chainok, K., Wannarit, N., Ruchirawat, S., and Thasana, N.

Journal of Organic Chemistry
Vol.: 86
No.: 14
Page: 9360-9383
Published: 2021
doi: https://doi.org/10.1021/acs.joc.1c00609

Identification of new 3-phenyl-1H-indole-2-carbohydrazide derivatives and their structure–activity relationships as potent tubulin inhibitors and anticancer agents: A combined in silico, in vitro and synthetic study

By: Saruengkhanphasit, R., Butkinaree, C., Ornnork, N., Lirdprapamongkol, K., Niwetmarin, W., Svasti, J., Ruchirawat, S., and Eurtivong, C.

Bioorganic Chemistry
Vol.: 110
No.:
Page:
Published: 2021
doi: https://doi.org/10.1016/j.bioorg.2021.104795

In Silico-Guided Rational Drug Design and Semi-synthesis of C(2)-Functionalized Huperzine A Derivatives as Acetylcholinesterase Inhibitors

By: Anukanon, S., Pongpamorn, P., Tiyabhorn, W., Chatwichien, J., Niwetmarin, W., Sessions, R. B., Ruchirawat, S., and Thasana, N.

ACS Omega
Vol.: 6
No.: 30
Page: 19924-19939
Published: 2021
doi: https://doi.org/10.1021/acsomega.1c02875

Investigations on Anticancer and Antimalarial Activities of Indole-Sulfonamide Derivatives and in Silico Studies

By: Pingaew, R., Mandi, P., Prachayasittikul, V., Thongnum, A., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.

ACS Omega
Vol.: 6
No.: 47
Page: 31854-31868
Published: 2021
doi: https://doi.org/10.1021/acsomega.1c04552

Isolation of Nucleic Acids Using Fly Ash as a Low-Cost Adsorbent

By: Thawornpan, P., Thanapongpichat, S., Tun, A. W., Jumpathong, W., Jong, L. D., and Buncherd, H.

Analytical Letters
Vol.: 54
No.: 12
Page: 2037-2050
Published: 2021
doi: https://doi.org/10.1080/00032719.2020.1835938

LC-QTOF-MS/MS based molecular networking approach for the isolation of α-glucosidase inhibitors and virucidal agents from coccinia grandis (L.) voigt

By: Astiti, M. A., Jittmittraphap, A., Leaungwutiwong, P., Chutiwitoonchai, N., Pripdeevech, P., Mahidol, C., Ruchirawat, S., and Kittakoop, P.

Foods
Vol.: 10
No.: 12
Page:
Published: 2021
doi: https://doi.org/10.3390/foods10123041

Magnetic Fraction of Fly Ash as a Low-Cost Magnetic Adsorbent for Selective Capture of Phosphoproteins

By: Thawornpan, P., Jumpathong, W., Thanapongpichat, S., Tansila, N., Win Tun, A., de Jong, L., and Buncherd, H.

Analytical Letters
Vol.: 54
No.: 11
Page: 1826-1839
Published: 2021
doi: https://doi.org/10.1080/00032719.2020.1825467

Microwave-Assisted Green Synthesis of 2,3-Dihydroquinazolinones under Base- and Catalyst-Free conditions

By: Kerdphon, S., Jongcharoenkamol, J., Chatwichien, J., Singh, T., Channei, D., Choommongkol, V., Rithchumpon, P., and Meepowpan, P.

Chemistryselect
Vol.: 6
No.: 19
Page: 4661-4669
Published: 2021
doi: https://doi.org/10.1002/slct.202101063

A New Bispyrroloiminoquinone Alkaloid From a Thai Collection of Clavelina sp

By: Grkovic, T., Ruchirawat, S., Kittakoop, P., Grothaus, P. G., Evans, J. R., Britt, J. R., Newman, D. J., Mahidol, C., and O’Keefe, B. R.

Asian Journal of Organic Chemistry
Vol.: 10
No.: 7
Page: 1647-1649
Published: 2021
doi: https://doi.org/10.1002/ajoc.202100155

NMR characterization of rearranged staurosporine aglycone analogues from the marine sponge Damiria sp

By: Tran, T. D., Cartner, L. K., Bokesch, H. R., Henrich, C. J., Wang, X. W., Mahidol, C., Ruchirawat, S., Kittakoop, P., O’Keefe, B. R., and Gustafson, K. R.

Magnetic Resonance in Chemistry
Vol.: 59
No.: 5
Page: 534-539
Published: 2021
doi: https://doi.org/10.1002/mrc.4932

Novel antimicrobial ciprofloxacin-pyridinium quaternary ammonium salts with improved physicochemical properties and DNA gyrase inhibitory activity

By: Ezelarab, H. A. A., Abbas, S. H., Abourehab, M. A. S., Badr, M., Sureram, S., Hongmanee, P., Kittakoop, P., Abuo-Rahma, G. E. D. A., and Hassan, H. A.

Medicinal Chemistry Research
Vol.: 30
No.: 12
Page: 2168-2183
Published: 2021
doi: https://doi.org/10.1007/s00044-021-02798-3

An optimised MALDI-TOF assay for phosphatidylcholine-specific phospholipase C

By: Sharma, N., Langley, R. J., Eurtivong, C., Leung, E., Dixon, R. J., Paulin, E. K., Rees, S. W. P., Pilkington, L. I., Barker, D., Reynisson, J., and Leung, I. K. H.

Analytical Methods
Vol.: 13
No.: 4
Page: 491-496
Published: 2021
doi: https://doi.org/10.1039/d0ay02208j

Oxazaborolidine-catalyzed reductive parallel kinetic resolution of ketones from β-nitro-azabicycles for the synthesis of chiral hypoestestatins 1, 2

By: Disadee, W., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 19
No.: 40
Page: 8794-8805
Published: 2021
doi: https://doi.org/10.1039/d1ob01608c

PdCl2-Catalyzed Oxidative Cyclization of N-(2’-Alkynylaryl)-1,3-ketoamides: Synthesis of 3,4-Diacyl-2-Quinolones

By: Punjajom, K., Tummatorn, J., Ruchirawat, S., and Thongsornkleeb, C.

Asian Journal of Organic Chemistry
Vol.: 10
No.: 4
Page: 906-917
Published: 2021
doi: https://doi.org/10.1002/ajoc.202100035

Roles of autophagy in relation to mitochondrial stress responses of HeLa cells to lamellarin cytotoxicity

By: Sopha, P., Phutubtim, N., Chantrathonkul, B., Ploypradith, P., Ruchirawat, S., and Chittchang, M.

Toxicology
Vol.: 462
No.:
Page:
Published: 2021
doi: https://doi.org/10.1016/j.tox.2021.152963

Separation of diethylpyrocarbonate-modified histidine-containing peptides using strong cation exchange chromatography

By: Thawonpan, P., Thanapongpichat, S., Jumpathong, W., Tun, A. W., Weeraphan, C., Wanitsuwan, W., and Buncherd, H.

Songklanakarin Journal of Science and Technology
Vol.: 43
No.: 5
Page: 1443-1448
Published: 2021
doi:

Spontaneous conversion of prenyl halides to acids: application in metal-free preparation of deuterated compounds under mild conditions

By: Darshana, D., Sureram, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.

Organic and Biomolecular Chemistry
Vol.: 19
No.: 34
Page: 7390-7402
Published: 2021
doi: https://doi.org/10.1039/d1ob01275d

Substituted 9-Anthraldehydes from Dibenzocycloheptanol Epoxides via Acid-Catalyzed Epoxide Opening/Semipinacol Rearrangement

By: Phumjan, T., Songthammawat, P., Jongcharoenkamol, J., Batsomboon, P., Ruchirawat, S., and Ploypradith, P.

Journal of Organic Chemistry
Vol.: 86
No.: 19
Page: 13322-13349
Published: 2021
doi: https://doi.org/10.1021/acs.joc.1c01405

Synthesis of Benzoazepine Derivatives via Azide Rearrangement and Evaluation of Their Antianxiety Activities

By: Reamtong, O., Lapmanee, S., Tummatorn, J., Palavong, N., Thongsornkleeb, C., and Ruchirawat, S.

ACS Medicinal Chemistry Letters
Vol.: 12
No.: 9
Page: 1449-1458
Published: 2021
doi: https://doi.org/10.1021/acsmedchemlett.1c00275

Synthesis of Isocryptolepine-Triazole Adducts and Evaluation of Their Cytotoxic Activity

By: Rodphon, W., Laohapaisan, P., Supantanapong, N., Reamtong, O., Ngiwsara, L., Lirdprapamongkol, K., Thongsornkleeb, C., Khunnawutmanotham, N., Tummatorn, J., Svasti, J., and Ruchirawat, S.

ChemMedChem
Vol.: 16
No.: 24
Page: 3750-3762
Published: 2021
doi: https://doi.org/10.1002/cmdc.202100554

Synthesis of sorafenib analogues incorporating a 1,2,3-triazole ring and cytotoxicity towards hepatocellular carcinoma cell lines

By: Palakhachane, S., Ketkaew, Y., Chuaypen, N., Sirirak, J., Boonsombat, J., Ruchirawat, S., Tangkijvanich, P., Suksamrarn, A., and Limpachayaporn, P.

Bioorganic Chemistry
Vol.: 112
No.:
Page:
Published: 2021
doi: https://doi.org/10.1016/j.bioorg.2021.104831

Synthesis, characterization and anticancer activity of Fe(II) and Fe(III) complexes containing N-(8-quinolyl)salicylaldimine Schiff base ligands

By: Wongsuwan, S., Chatwichien, J., Pinchaipat, B., Kumphune, S., Harding, D. J., Harding, P., Boonmak, J., Youngme, S., and Chotima, R.

Journal of Biological Inorganic Chemistry
Vol.: 26
No.: 2-3
Page: 327-339
Published: 2021
doi: https://doi.org/10.1007/s00775-021-01857-9

Total synthesis of microansamycin I

By: Sittihan, S., and Ruchirawat, S.

Tetrahedron Letters
Vol.: 68
No.:
Page:
Published: 2021
doi: https://doi.org/10.1016/j.tetlet.2021.152945

Utilization ofortho-alkynylarylcarbonyl derivatives for creating structurally diverse chemical compounds

By: Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 19
No.: 27
Page: 5982-5998
Published: 2021
doi: https://doi.org/10.1039/d1ob00629k

Uvarmicranones A and B, two new benzoquinones and cytotoxic constituents from the stems of Uvaria micrantha (A. DC.) Hook. f. & Thomson

By: Boonsombat, J., Thongnest, S., Kheawchaum, S., Mahidol, C., Ruchirawat, S., and Prawat, H.

Natural Product Research
Vol.: 35
No.: 24
Page: 5643-5652
Published: 2021
doi: https://doi.org/10.1080/14786419.2020.1824221

Visible-light-mediated decarboxylative alkylation of 2-pyridone derivatives: Via a C3-selective C-H functionalization

By: Niwetmarin, W., Saruengkhanphasit, R., Eurtivong, C., and Ruchirawat, S.

Organic and Biomolecular Chemistry
Vol.: 19
No.: 42
Page: 9231-9236
Published: 2021
doi: https://doi.org/10.1039/d1ob01829a

2020

Updated on January 28, 2021

1. An anticonvulsive drug, valproic acid (valproate), has effects on the biosynthesis of fatty acids and polyketides in microorganisms

By: Poolchanuan, P., Unagul, P., Thongnest, S., Wiyakrutta, S., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Scientific Reports
Vol.: 10
No.: 1
Page:
Published: 2020
doi: https://doi.org/10.1038/s41598-020-66251-y

2. Antifungal activity of 8-methoxynaphthalen-1-ol isolated from the endophytic fungus Diatrype palmicola MFLUCC 17-0313 against the plant pathogenic fungus Athelia rolfsii on tomatoes

By: Tanapichatsakul, C., Pansanit, A., Monggoot, S., Brooks, S., Prachya, S., Kittakoop, P., Panuwet, P., and Pripdeevech, P.
PeerJ
Vol.: 8
No.:
Page:
Published: 2020
doi: https://doi.org/10.7717/peerj.9103

3. Antioxidant and acetylcholinesterase inhibitory activities of Morinda citrifolia L. extracts

By: Sam-ang, P., Surangkul, D., Savaspun, K., and Phanumartwiwath, A.
Agriculture and Natural Resources
Vol.: 54
No.: 2
Page: 173–179
Published: 2020
doi:

4. Atalantiaphyllines A-G, prenylated acridones from Atalantia monophylla DC. and their aromatase inhibition and cytotoxic activities

By: Pailee, P., Prawat, H., Ploypradith, P., Mahidol, C., Ruchirawat, S., and Prachyawarakorn, V.
Phytochemistry
Vol.: 180
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.phytochem.2020.112525

5. Biscurcudiols, myrmekioperoxides, and myrmekiodermaral from the Thai marine sponge Myrmekioderma sp.

By: Wongbundit, S., Mahidol, C., Kaweetripob, W., Prachyawarakorn, V., Eurtivong, C., Sahakitpichan, P., Tuntiwachwuttikul, P., Ruchirawat, S., and Prawat, H.
Tetrahedron
Vol.: 76
No.: 19
Page:
Published: 2020
doi: https://doi.org/10.1016/j.tet.2020.131162

6. Chemoselective acid-catalyzed 4+2 -cycloaddition reactions of ortho-quinone methides and styrenes/stilbenes/cinnamates

By: Akkarasereenon, K., Tangdenpaisal, K., Ruchirawat, S., and Ploypradith, P.
Organic & Biomolecular Chemistry
Vol.: 18
No.: 43
Page: 8854-8866
Published: 2020
doi: https://doi.org/10.1039/d0ob01312a

7. Commercial Copper-Catalyzed Aerobic Oxidative Synthesis of Quinazolinones from 2-Aminobenzamide and Methanol

By: Kerdphon, S., Sanghong, P., Chatwichien, J., Choommongkol, V., Rithchumpon, P., Singh, T., and Meepowpan, P.
European Journal of Organic Chemistry
Vol.: 2020
No.: 18
Page: 2730-2734
Published: 2020
doi: https://doi.org/10.1002/ejoc.202000257

8. Discovery of New and Potent InhA Inhibitors as Antituberculosis Agents: Structure-Based Virtual Screening Validated by Biological Assays and X-ray Crystallography

By: Kamsri, P., Hanwarinroj, C., Phusi, N., Pornprom, T., Chayajarus, K., Punkvang, A., Suttipanta, N., Srimanote, P., Suttisintong, K., Songsiriritthigul, C., Saparpakorn, P., Hannongbua, S., Rattanabunyong, S., Seetaha, S., Choowongkomon, K., Sureram, S., Kittakoop, P., Hongmanee, P., Santanirand, P., Chen, Z. Q., Zhu, W. L., Blood, R. A., Takebayashi, Y., Hinchliffe, P., Mulholland, A. J., Spencer, J., and Pungpo, P.
Journal of Chemical Information and Modeling
Vol.: 60
No.: 1
Page: 226-234
Published: 2020
doi: https://doi.org/10.1021/acs.jcim.9b00918

9. Discovery of novel halogenated 8-hydroxyquinoline-based anti-MRSA agents: In vitro and QSAR studies

By: Cherdtrakulkiat, R., Worachartcheewan, A., Tantimavanich, S., Lawung, R., Sinthupoom, N., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Drug Development Research
Vol.: 81
No.: 1
Page: 127-135
Published: 2020
doi: https://doi.org/10.1002/ddr.21611

10. Discovery of novel phosphatidylcholine-specific phospholipase C drug-like inhibitors as potential anticancer agents

By: Eurtivong, C., Pilkington, L. I., van Rensburg, M., White, R. M., Brar, H. K., Rees, S., Paulin, E. K., Xu, C. S., Sharma, N., Leung, I. K. H., Leung, E., Barker, D., and Reynisson, J.
European Journal of Medicinal Chemistry
Vol.: 187
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.ejmech.2019.111919

11. Draft Genome Sequence of Diaporthe sp. Strain HANT25, an Endophytic Fungus Producing Mycoepoxydiene

By: Tulsook, K., Isarangkul, D., Sriubolmas, N., Kittakoop, P., and Wiyakrutta, S.
Microbiol Resour Announc
Vol.: 9
No.: 36
Page:
Published: 2020
doi: https://doi.org/10.1128/MRA.00805-20

12. First Draft Genome Sequence of Thermophilic Laceyella tengchongensis BKK01, Isolated from Municipal Solid Waste in Thailand

By: Wachiralurpan, S., Ruangsuj, P., Yamprayoonswat, W., Sopha, P., Jumpathong, W., Sittihan, S., Kanjanavas, P., Areekit, S., Chansiri, K., Chauyrod, K., and Yasawong, M.
Microbiology resource announcements
Vol.: 9
No.: 37
Page: 2
Published: 2020
doi: https://doi.org/10.1128/mra.00798-20

13. Functionalization at C2, C3, and C4 of quinolines: Discovery of water-soluble betaine dyes of C3 quinolinium derivatives with solvatochromic and pH-sensitive properties

By: Sangher, S., Kesornpun, C., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Dyes and Pigments
Vol.: 178
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.dyepig.2020.108341

14. Metal-Free, One-Pot Cascade Annulation of 2-Pyrones in Water for the Synthesis of Peptidomimetics

By: Disadee, W., Lekky, A., and Ruchirawat, S.
Journal of Organic Chemistry
Vol.: 85
No.: 4
Page: 1802-1822
Published: 2020
doi: https://doi.org/10.1021/acs.joc.9b01856

15. Molecular dynamics, MM/PBSA and in vitro validation of a novel quinazoline-based EGFR tyrosine kinase inhibitor identified using structure-based in silico screening

By: Ornnork, N., Kiriwan, D., Lirdprapamongkol, K., Choowongkomon, K., Svasti, J., and Eurtivong, C.
Journal of Molecular Graphics and Modelling
Vol.: 99
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.jmgm.2020.107639

16. Nickel Nanoparticle Catalyzed Mono- and Di-Reductions of gem-Dibromocyclopropanes Under Mild, Aqueous Micellar Conditions

By: Wood, A. B., Cortes-Clerget, M., Kincaid, J. R. A., Akkachairin, B., Singhania, V., Gallou, F., and Lipshutz, B. H.
Angew Chem Int Ed Engl
Vol.:
No.:
Page:
Published: 2020
doi: https://doi.org/10.1002/anie.202006162

17. Rapid synthesis of mycobacterial mannan polysaccharide with alkyne terminated linker

By: Bunthitsakda, W., Ruchirawat, S., and Boonyarattanakalin, S.
Suranaree Journal of Science and Technology
Vol.: 27
No.: 1
Page: 9
Published: 2020
doi:

18. Synthesis and antitumor activity of bis(arylsulfonyl)dihydroimidazolinone derivatives

By: Sittihan, S., Jumpathong, W., Sopha, P., and Ruchirawat, S.
Bioorganic and Medicinal Chemistry Letters
Vol.: 30
No.: 1
Page:
Published: 2020
doi: https://doi.org/10.1016/j.bmcl.2019.126776

19. Synthesis and neuroprotective effects of novel chalcone-triazole hybrids

By: Sooknual, P., Pingaew, R., Phopin, K., Ruankham, W., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Bioorganic Chemistry
Vol.: 105
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.bioorg.2020.104384

20. Synthesis of 4-Acylchromene via Highly Chemoselective Iodine-Catalyzed Cyclization of Alkynylarylether Dimethylacetals

By: Rodphon, W., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
Chemistry-an Asian Journal
Vol.: 15
No.: 21
Page: 3475-3486
Published: 2020
doi: https://doi.org/10.1002/asia.202000994

21. Synthesis of neocryptolepines and carbocycle-fused quinolines and evaluation of their anticancer and antiplasmodial activities

By: Akkachairin, B., Rodphon, W., Reamtong, O., Mungthin, M., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
Bioorganic Chemistry
Vol.: 98
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.bioorg.2020.103732

22. Synthesis, cytotoxicity evaluation, and molecular modeling studies of 2,N10-substituted acridones as DNA-intercalating agents

By: Khunnawutmanotham, N., Jumpathong, W., Eurtivong, C., Chimnoi, N., and Techasakul, S.
Journal of Chemical Research
Vol.: 44
No.: 7-8
Page: 410-425
Published: 2020
doi: https://doi.org/10.1177/1747519820902674

23. Transition-Metal-Catalyzed Suzuki-Miyaura-Type Cross-Coupling Reactions of pi-Activated Alcohols

By: Akkarasamiyo, S., Ruchirawat, S., Ploypradith, P., and Samec, J. S. M.
Synthesis-Stuttgart
Vol.: 52
No.: 5
Page: 645-659
Published: 2020
doi: https://doi.org/10.1055/s-0039-1690740

24. UHPLC-ESI-QTOF-MS/MS-Based Molecular Networking Guided Isolation and Dereplication of Antibacterial and Antifungal Constituents of Ventilago denticulata

By: Azizah, M., Pripdeevech, P., Thongkongkaew, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Antibiotics (Basel)
Vol.: 9
No.: 9
Page:
Published: 2020
doi: https://doi.org/10.3390/antibiotics9090606

2019

Updated on September 16, 2020

1. Draft Genome Sequence of Multidrug-Resistant Proteus mirabilis CKTH01, Isolated from Raw Chicken Meat

By: Areekit, S., Thongpramul, N., Yamprayoonswat, W., Jumpathong, W., Sittihan, S., Wanthongchareon, S., Ruangsuj, P., Wachiralurpan, S., Chansiri, K., and Yasawong, M.
Microbiology resource announcements
Vol.: 8
No.: 38
Page: e00861-00819
Published: 2019
doi: https://doi.org/10.1128/MRA.00861-19

2. A new 22, 26-seco physalin steroid from Physalis angulata

By: Boonsombat, J., Chawengrum, P., Mahidol, C., Kittakoop, P., Ruchirawat, S., and Thongnest, S.
Natural Product Research
Vol.: 34
No.: 8
Page: 1097-1104
Published: 2020
doi: https://doi.org/10.1080/14786419.2018.1550766

3. A Concise Approach to Oxo‐Dehydrorotenoid by Direct Lactonization and the Total Syntheses of Stemonone, Rotenonone, 6‐Oxo‐dehydroelliptone, and 6‐Oxo‐6a, 12a‐dehydrodeguelin

By: Boonsombat, J., Thongnest, S., and Ruchirawat, S.
European Journal of Organic Chemistry
Vol.: 2019
No.: 19
Page: 2971-2983
Published: 2019
doi: https://doi.org/10.1021/acs.orglett.5b02269

4. Serratene triterpenoids and their biological activities from Lycopodiaceae plants

By: Boonya-Udtayan, S., Thasana, N., Jarussophon, N., and Ruchirawat, S.
Fitoterapia
Vol.: 136
No.:
Page: 104181
Published: 2019
doi: https://doi.org/10.1016/j.fitote.2019.104181

5. Novel triazole-tetrahydroisoquinoline hybrids as human aromatase inhibitors

By: Chamduang, C., Pingaew, R., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Bioorganic Chemistry
Vol.: 93
No.:
Page: 103327
Published: 2019
doi: https://doi.org/10.1016/j.bioorg.2019.103327

6. Discovery of novel halogenated 8‐hydroxyquinoline‐based anti‐MRSA agents: In vitro and QSAR studies

7. Molecular docking study of lamellarin analogues and identification of potential inhibitors of HIV-1 integrase strand transfer complex by virtual screening

By: Eurtivong, C., Choowongkomon, K., Ploypradith, P., and Ruchirawat, S.
Heliyon
Vol.: 5
No.: 11
Page: e02811
Published: 2019
doi: https://doi.org/10.1016/j.heliyon.2019.e02811

8. The development of a weighted index to optimise compound libraries for high throughput screening

By: Eurtivong, C., and Reynisson, J.
Molecular Informatics
Vol.: 38
No.: 3
Page: 1800068
Published: 2019
doi: https://doi.org/10.1002/minf.201800068

9. Scandium (III)‐Triflate‐Catalyzed Pinacol‐Pinacolone Rearrangement and Cyclization of 1, 2‐Diaryl‐1, 2‐Ethanediol: A Versatile Synthesis of 1‐Aryl‐2, 3‐Dihydro‐1H‐3‐Benzazepines

By: Ieawsuwan, W., Pingaew, R., Kunkaewom, S., Ploypradith, P., and Ruchirawat, S.
Asian Journal of Organic Chemistry
Vol.: 8
No.: 8
Page: 1441-1447
Published: 2019
doi: https://doi.org/10.1002/ajoc.201900318

10. AN EFFICIENT SILVER TETRAFLUOROBORATE-CATALYZED CYCLOISOMERIZATION OF YNAMIDES (Dedicated to Professor Tohru Fukuyama on the occasion of his 70th birthday)

By: Ieawsuwan, W., and Ruchirawat, S.
Heterocycles: an international journal for reviews and communications in heterocyclic chemistry
Vol.: 99
No.: 1
Page: 100-110
Published: 2019
doi: https://doi.org/10.3987/COM-18-S(F)21

11. Exploitation of missing linker in Zr-based metal-organic framework as the catalyst support for selective oxidation of benzyl alcohol

By: Jumpathong, W., Pila, T., Lekjing, Y., Chirawatkul, P., Boekfa, B., Horike, S., and Kongpatpanich, K.
APL Materials
Vol.: 7
No.: 11
Page: 111109
Published: 2019
doi: https://doi.org/10.1063/1.5126077

12. In silico study directed towards identification of the key structural features of GyrB inhibitors targeting MTB DNA gyrase: HQSAR, CoMSIA and molecular dynamics simulations

By: Kamsri, P., Punkvang, A., Hannongbua, S., Suttisintong, K., Kittakoop, P., Spencer, J., Mulholland, A., and Pungpo, P.
SAR and QSAR in Environmental Research
Vol.: 30
No.: 11
Page: 775-800
Published: 2019
doi: https://doi.org/10.1080/1062936X.2019.1658218

13. Divergent Synthesis of 3-Hydroxyfluorene and 4-Azafluorene Derivatives from ortho-Alkynylarylketones

By: Laohapaisan, P., Chuangsoongnern, P., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
The Journal of organic chemistry
Vol.: 84
No.: 22
Page: 14451-14460
Published: 2019
doi: https://doi.org/10.1021/acs.joc.9b01825

14. Synthesis, molecular docking, and QSAR study of bis-sulfonamide derivatives as potential aromatase inhibitors

By: Leechaisit, R., Pingaew, R., Prachayasittikul, V., Worachartcheewan, A., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Bioorganic & Medicinal Chemistry
Vol.: 27
No.: 19
Page: 115040
Published: 2019
doi: https://doi.org/10.1016/j.bmc.2019.08.001

15. Rapid synthesis and immunogenicity of mycobacterial (1→ 5)-α-d-arabinofuranan

By: Leelayuwapan, H., Ruchirawat, S., and Boonyarattanakalin, S.
Carbohydrate Polymers
Vol.: 206
No.:
Page: 262-272
Published: 2019
doi: https://doi.org/10.1016/j.carbpol.2018.10.048

16. Stereoselective Convergent Synthesis of Tetrahydro-5 H-benzo [c] fluorene via Nine-Membered Ring-Closing Metathesis and Transannular Acid-Mediated Cyclization/Nucleophilic Addition

By: Lekky, A., Ruengsatra, T., Ruchirawat, S., and Ploypradith, P.
The Journal of organic chemistry
Vol.: 84
No.: 9
Page: 5277-5291
Published: 2019
doi: https://doi.org/10.1021/acs.joc.9b00263

17. The cytotoxic potential of cationic triangulenes against tumour cells

By: Leung, E., Pilkington, L. I., Naiya, M. M., Barker, D., Zafar, A., Eurtivong, C., and Reynisson, J.
MedChemComm
Vol.: 10
No.: 11
Page: 1881-1891
Published: 2019
doi: https://doi.org/10.1039/C9MD00305C

18. Construction of 5-Aminotetrazoles via in Situ Generation of Carbodiimidium Ions from Ketones Promoted by TMSN3/TfOH

By: Nimnual, P., Tummatorn, J., Boekfa, B., Thongsornkleeb, C., Ruchirawat, S., Piyachat, P., and Punjajom, K.
The Journal of organic chemistry
Vol.: 84
No.: 9
Page: 5603-5613
Published: 2019
doi: https://doi.org/10.1021/acs.joc.9b00555

19. Metal-Free Synthesis of 4-Chloroisocoumarins by TMSCl-Catalyzed NCS-Induced Chlorinative Annulation of 2-Alkynylaryloate Esters

By: Norseeda, K., Chaisan, N., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
The Journal of organic chemistry
Vol.: 84
No.: 24
Page: 16222-16236
Published: 2019
doi: https://doi.org/10.1021/acs.joc.9b02793

20. A Late-Stage Functionalization Approach to Derivatives of the Pyrano [3, 2-a] carbazole Natural Products

By: Norseeda, K., Gasser, V., and Sarpong, R.
The Journal of organic chemistry
Vol.: 84
No.: 9
Page: 5965-5973
Published: 2019
doi: https://doi.org/10.1021/acs.joc.9b00631

21. A novel potent autophagy inhibitor ECDD-S27 targets vacuolar ATPase and inhibits cancer cell survival

By: Paha, J., Kanjanasirirat, P., Munyoo, B., Tuchinda, P., Suvannang, N., Nantasenamat, C., Boonyarattanakalin, K., Kittakoop, P., Srikor, S., and Kongklad, G.
Scientific Reports
Vol.: 9
No.: 1
Page: 1-16
Published: 2019
doi: https://doi.org/10.1038/s41598-019-45641-x

22. Diverse flavonoids from the roots of Millettia brandisiana

By: Pailee, P., Mahidol, C., Ruchirawat, S., and Prachyawarakorn, V.
Phytochemistry
Vol.: 162
No.:
Page: 157-164
Published: 2019
doi: https://doi.org/10.1016/j.phytochem.2019.03.013

23. Rate Enhancement in CAN-Promoted Pd (PPh3) 2Cl2-Catalyzed Oxidative Cyclization: Synthesis of 2-Ketofuran-4-carboxylate Esters

By: Ruengsangtongkul, S., Chaisan, N., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
Organic Letters
Vol.: 21
No.: 8
Page: 2514-2517
Published: 2019
doi: https://doi.org/10.1021/acs.orglett.9b00053

24. Proteomic analysis of Plasmodium falciparum response to isocryptolepine derivative

By: Rujimongkon, K., Mungthin, M., Tummatorn, J., Ampawong, S., Adisakwattana, P., Boonyuen, U., and Reamtong, O.
PloS One
Vol.: 14
No.: 8
Page: e0220871
Published: 2019
doi: https://doi.org/10.1371/journal.pone.0220871

25. Synthetic Lipomannan Glycan Microarray Reveals the Importance of α (1, 2) Mannose Branching in DC-SIGN Binding

By: Sawettanai, N., Leelayuwapan, H., Karoonuthaisiri, N., Ruchirawat, S., and Boonyarattanakalin, S.
The Journal of organic chemistry
Vol.: 84
No.: 12
Page: 7606-7617
Published: 2019
doi: https://doi.org/10.1021/acs.joc.8b02944

26. Total Synthesis of the Marine Ladder Polyether Gymnocin B

By: Sittihan, S., and Jamison, T. F.
Journal of the American Chemical Society
Vol.: 141
No.: 28
Page: 11239-11244
Published: 2019
doi: https://doi.org/10.1021/jacs.9b04696

27. One-pot sequential synthesis of 3-carbonyl-4-arylbenzo [f] indole and 3-carbonyl-4-arylnaphthofuran fluorophores

By: Supantanapong, N., Chuangsoongnern, P., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
Organic Chemistry Frontiers
Vol.: 6
No.: 9
Page: 1340-1355
Published: 2019
doi: https://doi.org/10.1039/C8QO01182F

28. Total Synthesis of Palodesangren B Trimethyl Ether and D Dimethyl Ether via a Late-Stage Formation of 2 H-Pyran-2-one of the Tetrahydrobenzo [c] pyranochromenone Core

By: Tangdenpaisal, K., Songthammawat, P., Akkarasereenon, K., Chuayboonsong, K., Ruchirawat, S., and Ploypradith, P.
The Journal of organic chemistry
Vol.: 84
No.: 21
Page: 13410-13429
Published: 2019
doi: https://doi.org/10.1021/acs.joc.9b01596

29. Mechanistic investigation of phosphoprotein enrichment by fly ash-based chromatography

By: Thawornpan, P., Jumpathong, W., Thanapongpichat, S., de Jong, L., Phongdara, A., and Buncherd, H.
Journal of Chromatography B
Vol.: 1118
No.:
Page: 1-6
Published: 2019
doi: https://doi.org/10.1016/j.jchromb.2019.04.035

30. Vernodalidimer L, a sesquiterpene lactone dimer from Vernonia extensa and anti-tumor effects of vernodalin, vernolepin, and vernolide on HepG2 liver cancer cells

By: Thongnest, S., Chawengrum, P., Keeratichamroen, S., Lirdprapamongkol, K., Eurtivong, C., Boonsombat, J., Kittakoop, P., Svasti, J., and Ruchirawat, S.
Bioorganic Chemistry
Vol.: 92
No.:
Page: 103197
Published: 2019
doi: https://doi.org/10.1016/j.bioorg.2019.103197

31. Engineering faster transglycosidases and their acceptor specificity

By: Tran, L. T., Blay, V., Luang, S., Eurtivong, C., Choknud, S., González-Díaz, H., and Cairns, J. R. K.
Green Chemistry
Vol.: 21
No.: 10
Page: 2823-2836
Published: 2019
doi: https://doi.org/10.1039/C9GC00621D

32. NMR characterization of rearranged staurosporine aglycone analogues from the marine sponge Damiria sp

By: Tran, T. D., Cartner, L. K., Bokesch, H. R., Henrich, C. J., Wang, X. W., Mahidol, C., Ruchirawat, S., Kittakoop, P., O’Keefe, B. R., and Gustafson, K. R.
Magnetic Resonance in Chemistry
Vol.:
No.:
Page:
Published: 2019
doi: https://doi.org/10.1002/mrc.4932

33. Chemoselective Synthesis of 1, 1-Disubstituted Vinyl Triflates from Terminal Alkynes Using TfOH in the Presence of TMSN3

By: Tummatorn, J., Punjajom, K., Rodphon, W., Ruengsangtongkul, S., Chaisan, N., Lumyong, K., Thongsornkleeb, C., Nimnual, P., and Ruchirawat, S.
Organic Letters
Vol.: 21
No.: 12
Page: 4694-4697
Published: 2019
doi: https://doi.org/10.1021/acs.orglett.9b01576

34. Draft Genome Sequence of Haloferax volcanii SS0101, Isolated from Salt Farms in Samut Sakhon, Thailand

By: Wanthongcharoen, S., Yamprayoonswat, W., Ruangsuj, P., Thongpramul, N., Jumpathong, W., Sittihan, S., Kanjanavas, P., and Yasawong, M.
Microbiology resource announcements
Vol.: 8
No.: 46
Page:
Published: 2019
doi: https://doi.org/10.1128/MRA.00926-19

35. Draft Genome Sequence of Bacillus salarius IM0101, Isolated from Hypersaline Soil in Inner Mongolia, China

By: Yamprayoonswat, W., Boonvisut, S., Jumpathong, W., Sittihan, S., Ruangsuj, P., Wanthongcharoen, S., Thongpramul, N., Pimmason, S., Yu, B., and Yasawong, M.
Microbiology resource announcements
Vol.: 8
No.: 5
Page:
Published: 2019
doi: https://doi.org/10.1128/MRA.01686-18

36. Draft Genome Sequence of Thermophilic Halotolerant Aeribacillus pallidus TD1, Isolated from Tao Dam Hot Spring, Thailand

By: Yamprayoonswat, W., Sittihan, S., Jumpathong, W., and Yasawong, M.
Microbiology resource announcements
Vol.: 8
No.: 17
Page:
Published: 2019
doi: https://doi.org/10.1128/MRA.00204-19

37. Iridium-catalysed enantioselective formal deoxygenation of racemic alcohols via asymmetric hydrogenation

By: Zheng, J., Jongcharoenkamol, J., Peters, B. B., Guhl, J., Ponra, S., Ahlquist, M. S., and Andersson, P. G.
Nature Catalysis
Vol.: 2
No.: 12
Page: 1093-1100
Published: 2019
doi: https://doi.org/10.1038/s41929-019-0375-7

38. Evaluation of anti-tumour properties of two depsidones–Unguinol and Aspergillusidone D–in triple-negative MDA-MB-231 breast tumour cells

By: Zwartsen, A., Chottanapund, S., Kittakoop, P., Navasumrit, P., Ruchirawat, M., Van Duursen, M., and Van den Berg, M.
Toxicology Reports
Vol.: 6
No.:
Page: 1216-1222
Published: 2019
doi: https://doi.org/10.1016/j.toxrep.2019.10.012

39. Chemical synthesis of sulfated-α(1→6)-D-mannopyranan

By: Bunthitsakda, W., Wattanasiri, C., Somsak, R., and Siwarutt, B.
Songklanakarin Journal of Science & Technology
Vol.: 41
No.: 4
Page: 795-803
Published: 2019
doi:

2018

Updated on August 28, 2020

1. Domino N2-Extrusion–Cyclization of Alkynylarylketone Derivatives for the Synthesis of Indoloquinolines and Carbocycle-Fused Quinolines

By: Akkachairin, B., Tummatorn, J., Khamsuwan, N., Thongsornkleeb, C., and Ruchirawat, S.
The Journal of organic chemistry
Vol.: 83
No.: 18
Page: 11254-11268
Published: 2018
doi: https://doi.org/10.1021/acs.joc.8b01851

2. Controlled rapid synthesis and in vivo immunomodulatory effects of LM α (1, 6) mannan with an amine linker

By: Bunthitsakda, W., Leelayuwapan, H., Paha, J., Kangwanrangsan, N., Chawengkirttikul, R., Ponpuak, M., Ruchirawat, S., and Boonyarattanakalin, S.
Carbohydrate Polymers
Vol.: 195
No.:
Page: 420-431
Published: 2018
doi: https://doi.org/10.1016/j.carbpol.2018.04.045

3. PtCl4-catalyzed cyclization of N-acetyl-2-alkynylanilines: A mild and efficient synthesis of N-acetyl-2-substituted indoles

By: Chaisan, N., Kaewsri, W., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
Tetrahedron Letters
Vol.: 59
No.: 7
Page: 675-680
Published: 2018
doi: https://doi.org/10.1016/j.tetlet.2018.01.014

4. Cytotoxic and antimicrobial labdane and clerodane diterpenoids from Kaempferia elegans and Kaempferia pulchra

By: Chawengrum, P., Boonsombat, J., Kittakoop, P., Mahidol, C., Ruchirawat, S., and Thongnest, S.
Phytochemistry Letters
Vol.: 24
No.:
Page: 140-144
Published: 2018
doi: https://doi.org/10.1016/j.phytol.2018.02.009

5. One-pot cascade synthesis of azabicycles via the nitro-Mannich reaction and N-alkylation

By: Disadee, W., and Ruchirawat, S.
Organic & Biomolecular Chemistry
Vol.: 16
No.: 5
Page: 707-711
Published: 2018
doi: https://doi.org/10.1039/C7OB03104A

6. Selective divergent synthesis of indanols, indanones, and indenes via acid-mediated cyclization of (Z)-and (E)-(2-stilbenyl) methanols and its application for the synthesis of paucifloral F derivatives

By: Jongcharoenkamol, J., Chuathong, P., Amako, Y., Kono, M., Poonswat, K., Ruchirawat, S., and Ploypradith, P.
The Journal of organic chemistry
Vol.: 83
No.: 21
Page: 13184-13210
Published: 2018
doi: https://doi.org/10.1021/acs.joc.8b01921

7. Synthesis of 2‐Cyclohexenone‐2‐carboxylate and 4‐Chloro‐2‐cyclohexenone‐2‐carboxylate Derivatives by Cyclization of Alkyne‐Tethered 1, 3‐Ketoesters

By: Kaewsri, W., Norseeda, K., Ruengsangtongkul, S., Chaisan, N., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
Asian Journal of Organic Chemistry
Vol.: 7
No.: 1
Page: 203-211
Published: 2018
doi: https://doi.org/10.1002/ajoc.201700510

8. Cytotoxic sesterterpenes from thai marine sponge Hyrtios erectus

By: Kaweetripob, W., Mahidol, C., Tuntiwachwuttikul, P., Ruchirawat, S., and Prawat, H.
Marine Drugs
Vol.: 16
No.: 12
Page: 474
Published: 2018
doi: https://doi.org/10.3390/md16120474

9. Sesterterpenes and phenolic alkenes from the Thai sponge Hyrtios erectus

By: Kaweetripob, W., Mahidol, C., Wongbundit, S., Tuntiwachwuttikul, P., Ruchirawat, S., and Prawat, H.
Tetrahedron
Vol.: 74
No.: 2
Page: 316-323
Published: 2018
doi: https://doi.org/10.1016/j.tet.2017.11.073

10. Naphthalene derivatives and quinones from Ventilago denticulata and their nitric oxide radical scavenging, antioxidant, cytotoxic, antibacterial, and phosphodiesterase inhibitory activities

By: Molee, W., Phanumartwiwath, A., Kesornpun, C., Sureram, S., Ngamrojanavanich, N., Ingkaninan, K., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Chemistry & Biodiversity
Vol.: 15
No.: 3
Page: 1700537
Published: 2018
doi: https://doi.org/10.1002/cbdv.201700537

11. Three Lycopodium alkaloids from Thai club mosses

By: Nilsu, T., Thaisaeng, W., Thamnarak, W., Eurtivong, C., Jumraksa, A., Thorroad, S., Khunnawutmanotham, N., Ruchirawat, S., and Thasana, N.
Phytochemistry
Vol.: 156
No.:
Page: 83-88
Published: 2018
doi: https://doi.org/10.1016/j.phytochem.2018.09.001

12. Synthesis of β‐Naphthols and Naphthofuranones from ortho‐Alkynylarylketones via Sequential AgTFA‐Catalyzed Ketonization–Intramolecular Aldol Condensation: A Total Synthesis of Negundin A

By: Nimnual, P., Norseeda, K., Akkachairin, B., Tummatorn, J., Laohapaisan, P., Supantanapong, N., Chuangsoongnern, P., Thongsornkleeb, C., Sittihan, S., and Ruchirawat, S.
Asian Journal of Organic Chemistry
Vol.: 7
No.: 5
Page: 932-945
Published: 2018
doi: https://doi.org/10.1002/ajoc.201800025

13. Synthesis, molecular docking, and QSAR study of sulfonamide-based indoles as aromatase inhibitors

By: Pingaew, R., Mandi, P., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Medicinal Chemistry
Vol.: 143
No.:
Page: 1604-1615
Published: 2018
doi: https://doi.org/10.1016/j.ejmech.2017.10.057

14. Synthesis and molecular docking of N, N′-disubstituted thiourea derivatives as novel aromatase inhibitors

By: Pingaew, R., Prachayasittikul, V., Anuwongcharoen, N., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Bioorganic Chemistry
Vol.: 79
No.:
Page: 171-178
Published: 2018
doi: https://doi.org/10.1016/j.bioorg.2018.05.002

15. Semi-synthetic studies of α-onocerin derivatives for cytotoxicity

By: Pongpamorn, P., Wan-erlor, S., Ruchirawat, S., and Thasana, N.
Phytochemistry Letters
Vol.: 23
No.:
Page: 106-115
Published: 2018
doi: https://doi.org/10.1016/j.phytol.2017.11.017

16. Coriander (Coriandrum sativum): A promising functional food toward the well-being

By: Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Food Research International
Vol.: 105
No.:
Page: 305-323
Published: 2018
doi: https://doi.org/10.1016/j.foodres.2017.11.019

17. Base-mediated cascade cyclization: stereoselective synthesis of benzooxazocinone

By: Pramthaisong, C., Worayuthakarn, R., Pharikronburee, V., Duangthongyou, T., Rattanakam, R., Ruchirawat, S., and Thasana, N.
Organic Letters
Vol.: 20
No.: 13
Page: 4015-4019
Published: 2018
doi: https://doi.org/10.1021/acs.orglett.8b01573

18. A sensitive electrochemical immunosensor based on poly (2-aminobenzylamine) film modified screen-printed carbon electrode for label-free detection of human immunoglobulin G

By: Putnin, T., Jumpathong, W., Laocharoensuk, R., Jakmunee, J., and Ounnunkad, K.
Artificial cells, nanomedicine, and biotechnology
Vol.: 46
No.: 5
Page: 1042-1051
Published: 2018
doi: https://doi.org/10.1080/21691401.2017.1360322

19. Pd (II)-Ce (IV) cooperative induction of intramolecular oxidative cyclization of alpha-propargylated 1, 3-ketoesters: A rapid construction of 2, 4-diacylfurans

By: Ruengsangtongkul, S., Chaisan, N., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
2018 of Conference: 2018
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY: ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
Vol.: 256
No.:
Page:

20. Antagonistic activity against dirty panicle rice fungal pathogens and plant growth-promoting activity of Bacillus amyloliquefaciens BAS23

By: Saechow, S., Thammasittirong, A., Kittakoop, P., Prachya, S., and Thammasittirong, S. N.-R.
Journal of Microbiology and Biotechnology
Vol.: 28
No.: 9
Page: 1527-1535
Published: 2018
doi: https://doi.org/10.4014/jmb.1804.04025

21. Bioinspired Diastereoconvergent Synthesis of the Tricyclic Core of Palodesangrens via Diels–Alder Reaction, LiAlH4-Mediated Isomerization, and Acid-Mediated Cyclization

By: Songthammawat, P., Wangngae, S., Matsumoto, K., Duangkamol, C., Ruchirawat, S., and Ploypradith, P.
The Journal of organic chemistry
Vol.: 83
No.: 9
Page: 5225-5241
Published: 2018
doi: https://doi.org/10.1021/acs.joc.8b00668

22. The esterase B from Sphingobium sp. SM42 has the new de-arenethiolase activity against cephalosporin antibiotics

By: Sungkeeree, P., Toewiwat, N., Whangsuk, W., Ploypradith, P., Mongkolsuk, S., and Loprasert, S.
Biochemical and biophysical research communications
Vol.: 506
No.: 1
Page: 231-236
Published: 2018
doi: https://doi.org/10.1016/j.bbrc.2018.10.078

23. Synthesis of indoloquinolines via domino reactions of ortho-alkynylarylketones

By: Tummatorn, J., Akkachairin, B., Khamsuwan, N., Thongsornkleeb, C., and Ruchirawat, S.
2018 of Conference: 2018
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY: ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
Vol.: 256
No.:
Page:

24. Synthesis, antioxidant and antimicrobial activities of metal complexes of 2-thiouracil-hydroxyquinoline derivatives

By: Worachartcheewan, A., Pingaew, R., Lekcharoen, D., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Letters in Drug Design & Discovery
Vol.: 15
No.: 6
Page: 602-611
Published: 2018
doi: https://doi.org/10.2174/1570180814666170922163828

25. การประเมินปริมาณสารประกอบฟีนอลิกและเฟลโวนอยด์ในเมล็ดข้าวเพื่อการคัดเลือกสายพันธุ์ข้าวไทย (Oryza sativa L.)

By: สุธี ชุติไพจิตร, ธนวัช สุจริตวรกุล, และ ธณัฏฐ์คุณ มงคลอัศวรัตน์
วารสารวิชาการปทุมวัน
Vol.: 8
No.: 21
Page:
Published: 2018
doi:

2017

Updated on September 18, 2020

1. Silver-Catalyzed Cyclization of ortho-Carbonylarylacetylenols for the Synthesis of Dihydronaphthofurans

By: Akkachairin, B., Tummatorn, J., Supantanapong, N., Nimnual, P., Thongsornkleeb, C., and Ruchirawat, S.
Journal of Organic Chemistry
Vol.: 82
No.: 7
Page: 3727-3740
Published: 2017
doi: https://doi.org/10.1021/acs.joc.7b00198

2. First Vesicular Self-Assembly of Crotocembraneic Acid, a Nano-Sized Fourteen Membered Macrocyclic Diterpenic Acid

By: Bag, B. G., Barai, A. C., Wijesekera, K., and Kittakoop, P.
Chemistryselect
Vol.: 2
No.: 17
Page: 4969-4973
Published: 2017
doi: https://doi.org/10.1002/slct.201700500

3. First Hierarchical Self-Assembly of a Seco-Triterpenoid alpha-Onocerin Yielding Supramolecular Architectures

By: Bag, B. G., Hasan, S. K. N., Pongpamorn, P., and Thasana, N.
Chemistryselect
Vol.: 2
No.: 23
Page: 6650-6657
Published: 2017
doi: https://doi.org/10.1002/slct.201701285

4. Roscotanes and roscoranes: Oxygenated abietane and pimarane diterpenoids from Kaempferia roscoeana

By: Boonsombat, J., Mahidol, C., Chawengrum, P., Reuk-Ngam, N., Chimnoi, N., Techasakul, S., Ruchirawat, S., and Thongnest, S.
Phytochemistry
Vol.: 143
No.:
Page: 36-44
Published: 2017
doi: https://doi.org/10.1016/j.phytochem.2017.07.008

5. Superbanone, A New 2-Aryl-3-benzofuranone and Other Bioactive Constituents from the Tube Roots of Butea superba

By: Boonsombat, J., Prachyawarakorn, V., Pansanit, A., Mahidol, C., Ruchirawat, S., and Thongnest, S.
Chemistry & Biodiversity
Vol.: 14
No.: 7
Page:
Published: 2017
doi: https://doi.org/10.1002/cbdv.201700044

6. Iodine-Mediated Cyclization of ortho-Alkynylaryl Ketones for the Synthesis of Indenone Derivatives

By: Chuangsoongnern, P., Surinrach, C., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
European Journal of Organic Chemistry
Vol.: 2017
No.: 34
Page: 5102-5109
Published: 2017
doi: https://doi.org/10.1002/ejoc.201700968

7. A New Polyketide from the Endophytic Fungus Penicillium chermesinum

By: Darsih, C., Prachyawarakorn, V., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Indonesian Journal of Chemistry
Vol.: 17
No.: 3
Page: 360-364
Published: 2017
doi: https://doi.org/10.22146/ijc.22273

8. PIFA-BF3.OEt2 mediated intramolecular regioselective domino cyclization of ynamides: A novel method for the synthesis of tetrahydroisoquinoline-oxazol-2(3H)-ones

By: Ieawsuwan, W., and Ruchirawat, S.
Bioorganic & Medicinal Chemistry
Vol.: 25
No.: 11
Page: 2856-2867
Published: 2017
doi: https://doi.org/10.1016/j.bmc.2017.03.034

9. Homodimers of Vanillin and Apocynin Decrease the Metastatic Potential of Human Cancer Cells by Inhibiting the FAK/P13K/Akt Signaling Pathway

By: Jantaree, P., Lirdprapamongkol, K., Kaewsri, W., Thongsornkleeb, C., Choowongkomon, K., Atjanasuppat, K., Ruchirawatt, S., and Svasti, J.
Journal of Agricultural and Food Chemistry
Vol.: 65
No.: 11
Page: 2299-2306
Published: 2017
doi: https://doi.org/10.1021/acs.jafc.6b05697

10. A monoclonal antibody-based immunoassay for the determination of oxyresveratrol from Artocarpus lacucha Buch.-Ham

By: Kitisripanya, T., Inyai, C., Krittanai, S., Likhitwitayawuid, K., Sritularak, B., Ploypradith, P., Tanaka, H., Morimoto, S., and Putalun, W.
Journal of Natural Medicines
Vol.: 71
No.: 3
Page: 523-530
Published: 2017
doi: https://doi.org/10.1007/s11418-017-1083-8

11. Synthesis and Immunological Studies of the Lipomannan Backbone Glycans Found on the Surface of Mycobacterium tuberculosis

By: Leelayuwapan, H., Kangwanrangsan, N., Chawengkirttikul, R., Ponpuak, M., Charlermroj, R., Boonyarattanakalin, K., Ruchirawat, S., and Boonyarattanakalin, S.
Journal of Organic Chemistry
Vol.: 82
No.: 14
Page: 7190-7199
Published: 2017
doi: https://doi.org/10.1021/acs.joc.7b00703

12. Synthesis of phenanthridinones using Cu- or Pd-mediated C-N bond formation

By: Nealmongkol, P., Calmes, J., Ruchirawat, S., and Thasana, N.
Tetrahedron
Vol.: 73
No.: 6
Page: 735-741
Published: 2017
doi: https://doi.org/10.1016/j.tet.2016.12.051

13. Sterols from Thai Marine Sponge Petrosia (Strongylophora) sp and Their Cytotoxicity

By: Pailee, P., Mahidol, C., Ruchirawat, S., and Prachyawarakorn, V.
Marine Drugs
Vol.: 15
No.: 3
Page:
Published: 2017
doi: https://doi.org/10.3390/md15030054

14. Synthesis, biological evaluation and in silico study of bis-thiourea derivatives as anticancer, antimalarial and antimicrobial agents

By: Pingaew, R., Sinthupoom, N., Mandi, P., Prachayasittikul, V., Cherdtrakulkiat, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Medicinal Chemistry Research
Vol.: 26
No.: 12
Page: 3136-3148
Published: 2017
doi: https://doi.org/10.1007/s00044-017-2008-5

15. Roles of Pyridine and Pyrimidine Derivatives as Privileged Scaffolds in Anticancer Agents

By: Prachayasittikul, S., Pingaew, R., Worachartcheewan, A., Sinthupoom, N., Prachayasittikul, V., Ruchirawat, S., and Prachayasittikul, V.
Mini-Reviews in Medicinal Chemistry
Vol.: 17
No.: 10
Page: 869-901
Published: 2017
doi: https://doi.org/10.2174/1389557516666160923125801

16. AROMATASE INHIBITORY ACTIVITY OF 1,4-NAPHTHOQUINONE DERIVATIVES AND QSAR STUDY

By: Prachayasittikul, V., Pingaew, R., Worachartcheewan, A., Sitthimonchai, S., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 16
No.:
Page: 714-726
Published: 2017
doi: https://doi.org/10.17179/excli2017-309

17. A one-pot, metal-free approach to bicyclic 2-pyridones

By: Ruchirawat, S., and Disadee, W.
Organic Chemistry Frontiers
Vol.: 4
No.: 10
Page: 2026-2030
Published: 2017
doi: https://doi.org/10.1039/c7qo00406k

18. Antiplasmodial dimeric chalcone derivatives from the roots of Uvaria siamensis

By: Salae, A. W., Chairerk, O., Sukkoet, P., Chairat, T., Prawat, U., Tuntiwachwuttikul, P., Chalermglin, P., and Ruchirawat, S.
Phytochemistry
Vol.: 135
No.:
Page: 135-143
Published: 2017
doi: https://doi.org/10.1016/j.phytochem.2016.12.009

19. Copper Complexes of 8-Aminoquinoline and Uracils as Novel Aromatase Inhibitors

By: Sinthupoom, N., Prachayasittikul, V., Pingaew, R., Worachartcheewan, A., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Letters in Drug Design & Discovery
Vol.: 14
No.: 8
Page: 880-884
Published: 2017
doi: https://doi.org/10.2174/1570180813666161103144822

20. Divergent Strategy for the Diastereoselective Synthesis of the Tricyclic 6,7-Diaryltetrahydro-6H-benzo c chromene Core via Pt(IV)-Catalyzed Cycloaddition of o-Quinone Methides and Olefin Ring-Closing Metathesis

By: Tangdenpaisal, K., Chuayboonsong, K., Ruchirawat, S., and Ploypradith, P.
Journal of Organic Chemistry
Vol.: 82
No.: 5
Page: 2672-2688
Published: 2017
doi: https://doi.org/10.1021/acs.joc.6b03086

21. Ailanthusins A-G and nor-lupane triterpenoids from Ailanthus triphysa

By: Thongnest, S., Boonsombat, J., Prawat, H., Mahidol, C., and Ruchirawat, S.
Phytochemistry
Vol.: 134
No.:
Page: 98-105
Published: 2017
doi: https://doi.org/10.1016/j.phytochem.2016.11.007

22. Synthesis of synthetic mannan backbone polysaccharides found on the surface of Mycobacterium tuberculosis as a vaccine adjuvant and their immunological properties

By: Wattanasiri, C., Paha, J., Ponpuak, M., Ruchirawat, S., and Boonyarattanakalin, S.
Carbohydrate Polymers
Vol.: 175
No.:
Page: 746-755
Published: 2017
doi: https://doi.org/10.1016/j.carbpol.2017.07.045

23. Metabolite diversification by cultivation of the endophytic fungus Dothideomycete sp in halogen containing media: Cultivation of terrestrial fungus in seawater

By: Wijesekera, K., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Bioorganic & Medicinal Chemistry
Vol.: 25
No.: 11
Page: 2868-2877
Published: 2017
doi: https://doi.org/10.1016/j.bmc.2017.03.040

24. การตรวจสอบการเปลี่ยนแปลงการเจริญเติบโต รงควัตถุในการสังเคราะห์แสง และเอนไซม์ต้านอนุมูลอิสระในข้าวหอมที่ทดสอบด้วยวัสดุนาโนไทเทเนียมไดออกไซด์

By: สุธี ชุติไพจิตร, and ธณัฏฐ์คุณ มงคลอัศวรัตน์
วารสารวิชาการปทุมวัน
Vol.: 7
No.: 18
Page: 27-39
Published: 2017
doi:

2016

Updated on September 18, 2020

1. Oxyresveratrol: Structural Modification and Evaluation of Biological Activities

By: Chatsumpun, N., Chuanasa, T., Sritularak, B., Lipipun, V., Jongbunprasert, V., Ruchirawat, S., Ploypradith, P., and Likhitwitayawuid, K.
Molecules
Vol.: 21
No.: 4
Page:
Published: 2016
doi: https://doi.org/10.3390/molecules21040489

2. Derivatives (halogen, nitro and amino) of 8-hydroxyquinoline with highly potent antimicrobial and antioxidant activities

By: Cherdtrakulkiat, R., Boonpangrak, S., Sinthupoom, N., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Biochemistry and Biophysics Reports
Vol.: 6
No.:
Page: 135-141
Published: 2016
doi: https://doi.org/10.1016/j.bbrep.2016.03.014

3. Isomerizable (E/Z)-alkynyl-O-methyl oximes employing TMSCl-NCS in chlorinative cyclization for the direct synthesis of 4-chloroisoxazoles

By: Kaewsri, W., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
RSC Advances
Vol.: 6
No.: 54
Page: 48666-48675
Published: 2016
doi: https://doi.org/10.1039/c6ra09396e

4. Polyoxygenated ursane and oleanane triterpenes from Siphonodon celastrineus

By: Kaweetripob, W., Mahidol, C., Thongnest, S., Prawat, H., and Ruchirawat, S.
Phytochemistry
Vol.: 129
No.:
Page: 58-67
Published: 2016
doi: https://doi.org/10.1016/j.phytochem.2016.07.006

5. Water-Assisted Nitrile Oxide Cycloadditions: Synthesis of Isoxazoles and Stereoselective Syntheses of Isoxazolines and 1,2,4-Oxadiazoles

By: Kesornpun, C., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Angewandte Chemie-International Edition
Vol.: 55
No.: 12
Page: 3997-4001
Published: 2016
doi: https://doi.org/10.1002/anie.201511730

6. Optimizations of Hydroxyl Terminated Polymerization of Mannose Tricyclic Orthoester Toward Ready-to-use Lipomannan Backbone

By: Leelayuwapan, H., Ruchirawat, S., and Boonyarattanakalin, S.
Chiang Mai Journal of Science
Vol.: 43
No.: 1
Page: 1192-1200
Published: 2016
doi:

7. Squarrosine A and Pyrrolhuperzine A, New Lycopodium Alkaloids from Thai and Philippine Huperzia squarrosa

By: Nilsu, T., Thorroad, S., Ruchirawat, S., and Thasana, N.
Planta Medica
Vol.: 82
No.: 11-12
Page: 1046-1050
Published: 2016
doi: https://doi.org/10.1055/s-0042-106904

8. Streptanoate, a new anticancer butanoate from Streptomyces sp DC3

By: Noomnual, S., Thasana, N., Sungkeeree, P., Mongkolsuk, S., and Loprasert, S.
Journal of Antibiotics
Vol.: 69
No.: 2
Page: 124-127
Published: 2016
doi: https://doi.org/10.1038/ja.2015.95

9. Synthesis of 6-Alkyl-6H-benzo c chromene Derivatives by Cyclization/Selective Ether Cleavage in One Pot: Total Synthesis of Cannabinol

By: Norseeda, K., Tummatorn, J., Krajangsri, S., Thongsornkleeb, C., and Ruchirawat, S.
Asian Journal of Organic Chemistry
Vol.: 5
No.: 6
Page: 792-800
Published: 2016
doi: https://doi.org/10.1002/ajoc.201600095

10. ANTIMALARIAL AND ANTIMICROBIAL ACTIVITIES OF 8-AMINOQUINOLINE-URACILS METAL COMPLEXES

By: Phopin, K., Sinthupoom, N., Treeratanapiboon, L., Kunwittaya, S., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 15
No.:
Page: 144-152
Published: 2016
doi:

11. Lycoclavatumide and 8 beta,11 alpha-dihydroxylycopodine, a new fawcettimine and lycopodine-type alkaloid from Lycopodium clavatum

By: Pongpamorn, P., Wan-erlor, S., Ruchirawat, S., and Thasana, N.
Tetrahedron
Vol.: 72
No.: 44
Page: 7065-7069
Published: 2016
doi: https://doi.org/10.1016/j.tet.2016.09.046

12. Cytotoxic Steroidal Glycosides from the Whole Plant of Calamus acanthophyllus

By: Prawat, H., Mahidol, C., Kaweetripob, W., Intachote, P., Pisutjaroenpong, S., and Ruchirawat, S.
Planta Medica
Vol.: 82
No.: 11-12
Page: 1117-1121
Published: 2016
doi: https://doi.org/10.1055/s-0042-106972

13. Sesquiterpene isocyanides, isothiocyanates, thiocyanates, and formamides from the Thai sponge Halichondria sp

By: Prawat, H., Mahidol, C., Kaweetripob, W., Prachyawarakorn, V., Tuntiwachwuttikul, P., and Ruchirawat, S.
Tetrahedron
Vol.: 72
No.: 29
Page: 4222-4229
Published: 2016
doi: https://doi.org/10.1016/j.tet.2016.05.060

14. Effects of oxyresveratrol and its derivatives on cultured P19-derived neurons

By: Tadtong, S., Chatsumpun, N., Sritularak, B., Jongbunprasert, V., Ploypradith, P., and Likhitwitayawuid, K.
Tropical Journal of Pharmaceutical Research
Vol.: 15
No.: 12
Page: 2619-2628
Published: 2016
doi: https://doi.org/10.4314/tjpr.v15i12.12

15. Bacterial consortium expressing surface displayed, intra- and extracellular lipases and pseudopyronine B for the degradation of oil

By: Thiengmag, S., Chuencharoen, S., Thasana, N., Whangsuk, W., Jangiam, W., Mongkolsuk, S., and Loprasert, S.
International Journal of Environmental Science and Technology
Vol.: 13
No.: 8
Page: 2067-2078
Published: 2016
doi: https://doi.org/10.1007/s13762-016-1034-z

16. Cytotoxic sesquiterpenes from the endophytic fungus Pseudolagarobasidium acaciicola

By: Wibowo, M., Prachyawarakorn, V., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 122
No.:
Page: 126-138
Published: 2016
doi: https://doi.org/10.1016/j.phytochem.2015.11.016

17. A modified Cu(0)-Cu(I)-mediated C-aryl-C-aryl Ullmann coupling for the synthesis of biaryls

By: Yasamut, K., Jongcharoenkamol, J., Ruchirawat, S., and Ploypradith, P.
Tetrahedron
Vol.: 72
No.: 40
Page: 5994-6000
Published: 2016
doi: https://doi.org/10.1016/j.tet.2016.07.063

2015

Updated on September 18, 2020

1. Synthesis of isocryptolepine analogues and their structure-activity relationship studies as antiplasmodial and antiproliferative agents

By: Aroonkit, P., Thongsornkleeb, C., Tummatorn, J., Krajangsri, S., Mungthin, M., and Ruchirawat, S.
Eur J Med Chem
Vol.: 94
No.:
Page: 56-62
Published: 2015
doi: https://doi.org/10.1016/j.ejmech.2015.02.047

2. Optimization of microwave-assisted etherification of glycerol to polyglycerols by sodium carbonate as catalyst

By: Bookong, P., Ruchirawat, S., and Boonyarattanakalin, S.
Chemical Engineering Journal
Vol.: 275
No.:
Page: 253-261
Published: 2015
doi: https://doi.org/10.1016/j.cej.2015.04.033

3. Antimicrobial and cytotoxic acetogenin from Polyalthia debilis

By: Boonpangrak, S., Cherdtrakulkiat, R., Pingaew, R., Manam, P., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.

Journal of Applied Pharmaceutical Science
Vol.: 5
No.:
Page: 13-18
Published: 2015
doi: https://doi.org/10.7324/JAPS.2015.50303

4. Bioactive triterpenoids, antimicrobial, antioxidant and cytotoxic activities of Eclipta prostrata Linn

By: Cherdtrakulkiat, R., Boonpangrak, S., Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Journal of Applied Pharmaceutical Science
Vol.: 5
No.:
Page: 46-50
Published: 2015
doi: https://doi.org/10.7324/JAPS.2015.50308

5. Cytotoxic metabolites from the endophytic fungus Penicillium chermesinum: Discovery of a cysteine-targeted Michael acceptor as a pharmacophore for fragment-based drug discovery, bioconjugation and click reactions

By: Darsih, C., Prachyawarakorn, V., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
RSC Adv.
Vol.: 5
No.:
Page:
Published: 2015
doi: https://doi.org/10.1039/C5RA13735G

6. Antimycobacterial activity of natural products and synthetic agents: Pyrrolodiquinolines and vermelhotin as anti-tubercular leads against clinical multidrug resistant isolates of Mycobacterium tuberculosis

By: Ganihigama, D. U., Sureram, S., Sangher, S., Hongmanee, P., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
European Journal of Medicinal Chemistry
Vol.: 89
No.:
Page: 1-12
Published: 2015
doi: https://doi.org/10.1016/j.ejmech.2014.10.026

7. The Last and Next Decades of the Asian Core Program on Cutting-Edge Organic Chemistry in Asia

By: Isobe, M., Nishida, A., Choo, y.-m., Abd. Rahman, N., Ploypradith, P., Ruchirawat, S., Lin, G.-Q., Li, A., Yao, Z.-J., Uang, B.-J., Liao, C.-C., Chiu, P., Kim, B. M., and Loh, T.
Chemistry, an Asian Journal
Vol.: 10
No.:
Page: 790-804
Published: 2015
doi: https://doi.org/10.1002/asia.201500084

8. Cyclohexene long-chain fatty acid esters from Uvaria dulcis (Dunal)

By: Kaweetripob, W., Mahidol, C., Prawat, H., and Ruchirawat, S.
Phytochemistry Letters
Vol.: 12
No.:
Page: 248-251
Published: 2015
doi: https://doi.org/10.1016/j.phytol.2015.04.020

9. Chapter 5. Anticancer Drugs and Potential Anticancer Leads Inspired by Natural Products

By: Kittakoop, P.
Studies in Natural Products Chemistry
Vol.: 44
No.:
Page: 251-307
Published: 2015
doi: https://doi.org/10.1016/B978-0-444-63460-3.00005-5

10. Drimane Sesquiterpene-Conjugated Amino Acids from a Marine Isolate of the Fungus Talaromyces minioluteus (Penicillium Minioluteum)

By: Ngokpol, S., Suwakulsiri, W., Sureram, S., Lirdprapamongkol, K., Aree, T., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Marine Drugs
Vol.: 13
No.: 6
Page: 3567-3580
Published: 2015
doi: https://doi.org/10.3390/md13063567

11. Utility of Nitrogen Extrusion of Azido Complexes for the Synthesis of Nitriles, Benzoxazoles, and Benzisoxazoles

By: Nimnual, P., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
The Journal of organic chemistry
Vol.: 80
No.: 17
Page: 8657-8667
Published: 2015
doi: https://doi.org/10.1021/acs.joc.5b01305

12. Bioactive cardinane sesquiterpenes from the stems of Alangium salviifolium

By: Pailee, P., Prachyawarakorn, V., Ruchirawat, S., and Mahidol, C.
Chemistry, an Asian Journal
Vol.: 10
No.: 4
Page: 910-914
Published: 2015
doi: https://doi.org/10.1002/asia.201403253

13. Cytotoxic and cancer chemopreventive properties of prenylated stilbenoids from Macaranga siamensis

By: Pailee, P., Sangpetsiripan, S., Mahidol, C., Ruchirawat, S., and Prachyawarakorn, V.
Tetrahedron
Vol.: 71
No.: 34
Page: 5562-5571
Published: 2015
doi: https://doi.org/10.1016/j.tet.2015.06.058

14. 5-Methyl ether flavone glucosides from the leaves of Bruguiera gymnorrhiza

By: Panyadee, A., Sahakitpichan, P., Ruchirawat, S., and Kanchanapoom, T.
Phytochemistry Letters
Vol.: 11
No.:
Page: 215-219
Published: 2015
doi: https://doi.org/10.1016/j.phytol.2014.12.021

15. Synthesis and molecular docking of 1,2,3-triazole-based sulfonamides as aromatase inhibitors

By: Pingaew, R., Prachayasittikul, V., Mandi, P., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Bioorganic & Medicinal Chemistry
Vol.: 23
No.: 13
Page: 3472-3480
Published: 2015
doi: https://doi.org/10.1016/j.bmc.2015.04.036

16. Novel 1,4-naphthoquinone-based sulfonamides: Synthesis, QSAR, anticancer and antimalarial studies

By: Pingaew, R., Prachayasittikul, V., Worachartcheewan, A., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Medicinal Chemistry
Vol.: 103
No.:
Page: 446-459
Published: 2015
doi: https://doi.org/10.1016/j.ejmech.2015.09.001

17. Discovery of novel 1,2,3-triazole derivatives as anticancer agents using QSAR and in silico structural modification

By: Prachayasittikul, V., Pingaew, R., Anuwongcharoen, N., Worachartcheewan, A., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
SpringerPlus
Vol.: 4
No.:
Page: 571-571
Published: 2015
doi: https://doi.org/10.1186/s40064-015-1352-5

18. Glucosides of phenylpropanoic acid derivatives and coumarins from Micromelum minutum

By: Sahakitpichan, P., Tanpatanan, W., Chimnoi, N., Ruchirawat, S., and Kanchanapoom, T.
Phytochemistry Letters
Vol.: 14
No.:
Page: 12-16
Published: 2015
doi: https://doi.org/10.1016/j.phytol.2015.08.009

19. Nicotinic acid and derivatives as multifunctional pharmacophores for medical applications

By: Sinthupoom, N., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
European Food Research and Technology
Vol.: 240
No.: 1
Page: 1-17
Published: 2015
doi: https://doi.org/10.1007/s00217-014-2354-1

20. Synthesis of C4 – C5 cycloalkyl-fused and C6-modified chromans via ortho-quinone methides

By: Tangdenpaisal, K., Chuayboonsong, K., Sukjarean, P., Katesampao, V., Noiphrom, N., Ruchirawat, S., and Ploypradith, P.
Chemistry, an Asian Journal
Vol.: 10
No.: 4
Page: 1050-1064
Published: 2015
doi: https://doi.org/10.1002/asia.201403356

21. Designing new analogs for streamlining the structure of cytotoxic lamellarin natural products

By: Tangdenpaisal, K., Worayuthakarn, R., Karnkla, S., Ploypradith, P., Intachote, P., Sengsai, S., Saimanee, B., Ruchirawat, S., and Chittchang, M.
Chemistry, an Asian Journal
Vol.: 10
No.: 4
Page: 925-937
Published: 2015
doi: https://doi.org/10.1002/asia.201403361

22. Facile and Divergent Synthesis of Lamellarins and Lactam-Containing Derivatives with Improved Drug Likeness and Biological Activities

By: Theppawong, A., Ploypradith, P., Chuawong, P., Ruchirawat, S., and Chittchang, M.
Chemistry, an Asian Journal
Vol.: 10
No.: 12
Page: 2631-2650
Published: 2015
doi: https://doi.org/10.1002/asia.201500611

23. Regioselective Synthesis of 3-Bromoquinoline Derivatives and Diastereoselective Synthesis of Tetrahydroquinolines via Acid-Promoted Rearrangement of Arylmethyl Azides

By: Tummatorn, J., Poonsilp, P., Nimnual, P., Janprasit, J., Thongsornkleeb, C., and Ruchirawat, S.
The Journal of organic chemistry
Vol.: 80
No.: 9
Page: 4516-4525
Published: 2015
doi: https://doi.org/10.1021/acs.joc.5b00375

24. Convenient and Direct Azidation of sec-Benzyl Alcohols by Trimethylsilyl Azide with Bismuth(III) Triflate Catalyst

By: Tummatorn, J., Thongsornkleeb, C., Ruchirawat, S., Thongaram, P., and Kaewmee, B.
Synthesis
Vol.: 47
No.: 03
Page: 323-329
Published: 2015
doi: https://doi.org/10.1055/s-0034-1379967

25. Antimicrobial, antioxidant and anticancer activities of Strychnos lucida R. Br

By: Worachartcheewan, A., Sarmento, N., Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
African Journal of Traditional, Complementary and Alternative Medicines
Vol.: 12
No.:
Page: 122-127
Published: 2015
doi: https://doi.org/10.4314/ajtcam.v12i4.3042

2014

Updated on September 18, 2020

1. α-Glucosidase inhibitory activities of isoflavanones, isoflavones, and pterocarpans from Mucuna pruriens

By: Dendup, T., Prachyawarakorn, V., Pansanit, A., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Planta Medica
Vol.: 80
No.: 7
Page: 604-608
Published: 2014
doi: https://doi.org/10.1055/s-0034-1368427

2. One strain-many compounds (OSMAC) method for production of polyketides, azaphilones, and an isochromanone using the endophytic fungus Dothideomycete sp

By: Hewage, R. T., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 108
No.:
Page: 87-94
Published: 2014
doi: https://doi.org/10.1016/j.phytochem.2014.09.013

3. JSPS Asian Core Program: 7th & 8th ICCEOCA (Phase II/NICCEOCA-3 & -4), 2nd & 3rd Junior ICCEOCA, and Partly IUPAC Asian Project

By: Isobe, M., Murata, M., Hanashima, S., Nishida, A., Loh, T. P., Rahman, N. A., Thasana, N., and Chittchang, M.
Chemistry – An Asian Journal
Vol.: 9
No.: 7
Page: 1689-1696
Published: 2014
doi: https://doi.org/10.1002/asia.201402189

4. Alkaloids as important scaffolds in therapeutic drugs for the treatments of cancer, tuberculosis, and smoking cessation

By: Kittakoop, P., Mahidol, C., and Ruchirawat, S.
Current Topics in Medicinal Chemistry
Vol.: 14
No.: 2
Page: 239-252
Published: 2014
doi: https://doi.org/10.2174/1568026613666131216105049

5. Recent investigations of bioactive natural products from endophytic, marine-derived, insect pathogenic fungi and Thai medicinal plants

By: Mahidol, C., Kittakoop, P., Prachyawarakorn, V., Pailee, P., Prawat, H., and Ruchirawat, S.
Pure and Applied Chemistry
Vol.: 86
No.: 6
Page: 979
Published: 2014
doi: https://doi.org/10.1515/pac-2013-1206

6. Practical and Metal-Free Electrophilic Aromatic Halogenation by Interhalogen Compounds Generated In Situ from N-Halosuccinimide and Catalytic TMSCl

By: Maibunkaew, T., Thongsornkleeb, C., Tummatorn, J., Bunrit, A., and Ruchirawat, S.
Synlett
Vol.: 25
No.:
Page: 1769-1775
Published: 2014
doi: https://doi.org/10.1055/s-0034-1378225

7. Design, synthesis and molecular docking studies of novel N-benzenesulfonyl-1,2,3,4-tetrahydroisoquinoline-based triazoles with potential anticancer activity

By: Pingaew, R., Mandi, P., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Medicinal Chemistry
Vol.: 81
No.:
Page: 192-203
Published: 2014
doi: https://doi.org/10.1016/j.ejmech.2014.05.019

8. Synthesis and cytotoxicity of novel 4-(4-(substituted)-1H-1,2,3-triazol-1-yl)-N-phenethylbenzenesulfonamides

By: Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Medicinal Chemistry Research
Vol.: 23
No.: 4
Page: 1768-1780
Published: 2014
doi: https://doi.org/10.1007/s00044-013-0777-z

9. Synthesis, biological evaluation and molecular docking of novel chalcone-coumarin hybrids as anticancer and antimalarial agents

By: Pingaew, R., Saekee, A., Mandi, P., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Eur J Med Chem
Vol.: 85
No.:
Page: 65-76
Published: 2014
doi: https://doi.org/10.1016/j.ejmech.2014.07.087

10. Investigation of aromatase inhibitory activity of metal complexes of 8-hydroxyquinoline and uracil derivatives

By: Prachayasittikul, V., Pingaew, R., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Drug Design, Development and Therapy
Vol.: 8
No.:
Page: 1089-1096
Published: 2014
doi: https://doi.org/10.2147/DDDT.S67300

11. Synthesis, anticancer activity and QSAR study of 1,4-naphthoquinone derivatives

By: Prachayasittikul, V., Pingaew, R., Worachartcheewan, A., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Medicinal Chemistry
Vol.: 84
No.:
Page: 247-263
Published: 2014
doi: https://doi.org/10.1016/j.ejmech.2014.07.024

12. New trans- and cis-p-coumaroyl flavonol tetraglycosides from the leaves of Mitragyna rotundifolia

By: Sahakitpichan, P., Chadmuk, P., Disadee, W., Chimnoi, N., Ruchirawat, S., and Kanchanapoom, T.
Phytochemistry Letters
Vol.: 8
No.:
Page: 65-68
Published: 2014
doi: https://doi.org/10.1016/j.phytol.2014.02.002

13. An organocatalyst from renewable materials for the synthesis of coumarins and chromenes: Three-component reaction and multigram scale synthesis

By: Sangsuwan, R., Sangher, S., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
RSC Advances
Vol.: 4
No.:
Page: 13708-13718
Published: 2014
doi: https://doi.org/10.1039/c4ra00673a

14. Synthesis of the thyroid hormone analog GC-1 via Bi(OTf)3-catalyzed benzylation

By: Tangdenpaisal, K., Ruchirawat, S., and Ploypradith, P.
Tetrahedron
Vol.: 70
No.: 38
Page: 6789-6795
Published: 2014
doi: /https://doi.org/10.1016/j.tet.2014.07.063

15. Three new Lycopodium alkaloids from Huperzia carinata and Huperzia squarrosa

By: Thorroad, S., Worawittayanont, P., Khunnawutmanotham, N., Chimnoi, N., Jumruksa, A., Ruchirawat, S., and Thasana, N.
Tetrahedron
Vol.: 70
No.: 43
Page: 8017-8022
Published: 2014
doi: https://doi.org/10.1016/j.tet.2014.08.042

16. ZrCl4-promoted facile synthesis of indole derivatives

By: Tummatorn, J., Gleeson, M. P., Krajangsri, S., Thongsornkleeb, C., and Ruchirawat, S.
RSC Advances
Vol.: 4
No.: 38
Page: 20048-20052
Published: 2014
doi: https://doi.org/10.1039/C4RA02158D

17. A new synthetic approach to 6-unsubstituted phenanthridine and phenanthridine-like compounds under mild and metal-free conditions

By: Tummatorn, J., Krajangsri, S., Norseeda, K., Thongsornkleeb, C., and Ruchirawat, S.
Organic & Biomolecular Chemistry
Vol.: 12
No.: 28
Page: 5077-5081
Published: 2014
doi: https://doi.org/10.1039/c4ob00797b

18. Allyl 3, 4, 6-Tri-O-Benzyl-α-D-Mannopyranoside

By: Wattanasiri, C., Ruchirawat, S., Platon, M., and Boonyarattanakalin, S.
Carbohydrate Chemistry
Vol.:
No.:
Page: 188-193
Published: 2014
doi:

19. Tricyclic and Spirobicyclic Norsesquiterpenes from the Endophytic Fungus Pseudolagarobasidium acaciicola

By: Wibowo, M., Prachyawarakorn, V., Aree, T., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
European Journal of Organic Chemistry
Vol.: 2014
No.: 19
Page: 3976-3980
Published: 2014
doi: https://doi.org/10.1002/ejoc.201402262

20. Terpenoids from the roots of Drypetes hoaensis and their cytotoxic activities

By: Wittayalai, S., Mahidol, C., Prachyawarakorn, V., Prawat, H., and Ruchirawat, S.
Phytochemistry
Vol.: 99
No.:
Page: 121-126
Published: 2014
doi: https://doi.org/10.1016/j.phytochem.2013.12.017

21. Total Synthesis of Unsymmetrical Benzils, Scandione and Calophione A

By: Worayuthakarn, R., Boonya-udtayan, S., Ruchirawat, S., and Thasana, N.
European Journal of Organic Chemistry
Vol.: 2014
No.: 12
Page: 2496-2507
Published: 2014
doi: https://doi.org/10.1002/ejoc.201301722

22. Controlled ring-opening polymerization of 1,2,6-tricyclic orthoesters of mannose toward size-controlled alpha-D-mannopyranan

By: Yongyat, C., Ruchirawat, S., and Boonyarattanakalin, S.
E-Polymers
Vol.: 14
No.:
Page: 383-390
Published: 2014
doi: https://doi.org/10.1515/epoly-2014-0129

2013

Updated on September 18, 2020

1. Chemical constituents of Thai propolis

By: Athikomkulchai, S., Awale, S., Ruangrungsi, N., Ruchirawat, S., and Kadota, S.
Fitoterapia
Vol.: 88
No.:
Page: 96-100
Published: 2013
doi: https://doi.org/10.1016/j.fitote.2013.04.008

2. DBU-mediated regioselective intramolecular cyclization/dehydration of ortho diketo phenoxyethers: a synthesis of 2,3-substituted γ-benzopyranones

By: Bensulong, S., Boonsombat, J., and Ruchirawat, S.
Tetrahedron
Vol.: 69
No.: 44
Page: 9335-9348
Published: 2013
doi: https://doi.org/10.1016/j.tet.2013.07.104

3. Ring opening polymerization of mannosyl tricyclic orthoesters: rationalising the stereo and regioselectivity of glycosidic bond formation using quantum chemical calculations

By: Boonyarattanakalin, S., Ruchirawat, S., and Gleeson, M. P.
MedChemComm
Vol.: 4
No.: 1
Page: 265-268
Published: 2013
doi: https://doi.org/10.1039/C2MD20178J

4. Crystal Structure of 2-(2-Carboxy-4-hydroxy-6-methoxyphenoxy)-3, 5-dichloro-6-hydroxy-4-methylbenzoic Acid 1-Methyl Ester

By: Jongrungruangchok, S., Aree, T., Sureram, S., and Kittakoop, P.
Jiegou Huaxue
Vol.: 32
No.: 11
Page: 1742-1748
Published: 2013
doi:

5. Lupane, friedelane, oleanane, and ursane triterpenes from the stem of Siphonodon celastrineus Griff

By: Kaweetripob, W., Mahidol, C., Prawat, H., and Ruchirawat, S.
Phytochemistry
Vol.: 96
No.:
Page: 404-417
Published: 2013
doi: https://doi.org/10.1016/j.phytochem.2013.09.027

6. Synthesis of integerrimide A by an on-resin tandem Fmoc-deprotection-macrocyclisation approach

By: Kumarn, S., Chimnoi, N., and Ruchirawat, S.
Organic & Biomolecular Chemistry
Vol.: 11
No.: 44
Page: 7760-7767
Published: 2013
doi: https://doi.org/10.1039/c3ob41447g

7. Chrysin overcomes TRAIL resistance of cancer cells through Mcl-1 downregulation by inhibiting STAT3 phosphorylation

By: Lirdprapamongkol, K., Sakurai, H., Abdelhamed, S., Yokoyama, S., Athikomkulchai, S., Viriyaroj, A., Awale, S., Ruchirawat, S., Svasti, J., and Saiki, I.
International Journal of Oncology
Vol.: 43
No.: 1
Page: 329-337
Published: 2013
doi: https://doi.org/10.3892/ijo.2013.1926

8. A flavonoid chrysin suppresses hypoxic survival and metastatic growth of mouse breast cancer cells

By: Lirdprapamongkol, K., Sakurai, H., Abdelhamed, S., Yokoyama, S., Maruyama, T., Athikomkulchai, S., Viriyaroj, A., Awale, S., Yagita, H., Ruchirawat, S., Svasti, J., and Saiki, I.
Oncology Reports
Vol.: 30
No.: 5
Page: 2357-2364
Published: 2013
doi: https://doi.org/10.3892/or.2013.2667

9. Cu(I)-mediated lactone formation in subcritical water: a benign synthesis of benzopyranones and urolithins A–C

By: Nealmongkol, P., Tangdenpaisal, K., Sitthimonchai, S., Ruchirawat, S., and Thasana, N.
Tetrahedron
Vol.: 69
No.: 44
Page: 9277-9283
Published: 2013
doi: https://doi.org/10.1016/j.tet.2013.08.045

10. Vermelhotin, an Anti-inflammatory Agent, Suppresses Nitric Oxide Production in RAW 264.7 Cells via p38 Inhibition

By: Pansanit, A., Park, E.-J., Kondratyuk, T. P., Pezzuto, J. M., Lirdprapamongkol, K., and Kittakoop, P.
Journal of Natural Products
Vol.: 76
No.: 9
Page: 1824-1827
Published: 2013
doi: https://doi.org/10.1021/np400565e

11. Phenylethanoid and flavone glycosides from Ruellia tuberosa L

By: Phakeovilay, C., Disadee, W., Sahakitpichan, P., Sitthimonchai, S., Kittakoop, P., Ruchirawat, S., and Kanchanapoom, T.
Journal of Natural Medicines
Vol.: 67
No.: 1
Page: 228-233
Published: 2013
doi: https://doi.org/10.1007/s11418-012-0658-7

12. Synthesis and cytotoxicity of novel N-sulfonyl-1,2,3,4-tetrahydroisoquinoline thiosemicarbazone derivatives

By: Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Medicinal Chemistry Research
Vol.: 22
No.: 1
Page: 267-277
Published: 2013a
doi: https://doi.org/10.1007/s00044-012-0025-y

13. Synthesis and structure–activity relationship of mono-indole-, bis-indole-, and tris-indole-based sulfonamides as potential anticancer agents

By: Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Molecular Diversity
Vol.: 17
No.:
Page:
Published: 2013b
doi: https://doi.org/10.1007/s11030-013-9457-7

14. Tungstophosphoric acid catalyzed synthesis of N-sulfonyl-1,2,3,4-tetrahydroisoquinoline analogs

By: Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Chinese Chemical Letters
Vol.: 24
No.: 10
Page: 941-944
Published: 2013c
doi: https://doi.org/10.1016/j.cclet.2013.06.019

15. Cytotoxicity and QSAR study of (thio)ureas derived from phenylalkylamines and pyridylalkylamines

By: Pingaew, R., Tongraung, P., Worachartcheewan, A., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Medicinal Chemistry Research
Vol.: 22
No.:
Page:
Published: 2013
doi: https://doi.org/10.1007/s00044-012-0402-6

16. Synthesis, cytotoxicity and QSAR study of N-tosyl-1,2,3,4-tetrahydroisoquinoline derivatives

By: Pingaew, R., Worachartcheewan, A., Nantasenamat, C., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Archives of Pharmacal Research
Vol.: 36
No.: 9
Page: 1066-1077
Published: 2013
doi: https://doi.org/10.1007/s12272-013-0111-9

17. Transition Metal Complexes of 8-Aminoquinoline-5-Substituted Uracils with Antioxidative and Cytotoxic Activities

By: Pingaew, R., Worachartcheewan, A., Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Letters in Drug Design & Discovery
Vol.: 10
No.:
Page: 859-864
Published: 2013
doi: https://doi.org/10.2174/15701808113109990004

18. 8-Hydroxyquinolines: a review of their metal chelating properties and medicinal applications

By: Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Drug Design, Development and Therapy
Vol.: 7
No.:
Page: 1157-1178
Published: 2013a
doi: https://doi.org/10.2147/DDDT.S49763

19. High therapeutic potential of Spilanthes acmella: A review

By: Prachayasittikul, V., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 12
No.:
Page: 291-312
Published: 2013b
doi:

20. Flavans from Desmos cochinchinensis as potent aromatase inhibitors

By: Prachyawarakorn, V., Sangpetsiripan, S., Surawatanawong, P., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
MedChemComm
Vol.: 4
No.: 12
Page: 1590-1596
Published: 2013
doi: https://doi.org/10.1039/C3MD00166K

21. Glucopyranosyloxybenzyl derivatives of (R)-2-benzylmalic acid and (R)-eucomic acid, and an aromatic glucoside from the pseudobulbs of Grammatophyllum speciosum

By: Sahakitpichan, P., Mahidol, C., Disadee, W., Chimnoi, N., Ruchirawat, S., and Kanchanapoom, T.
Tetrahedron
Vol.: 69
No.: 3
Page: 1031-1037
Published: 2013
doi: https://doi.org/10.1016/j.tet.2012.11.082

22. Synthesis of Substituted 2-Arylindanes from E-(2-Stilbenyl)methanols via Lewis Acid-Mediated Cyclization and Nucleophililc Transfer from Trialkylsilyl Reagents

By: Sarnpitak, P., Trongchit, K., Kostenko, Y., Sathalalai, S., Gleeson, M. P., Ruchirawat, S., and Ploypradith, P.
The Journal of organic chemistry
Vol.: 78
No.: 17
Page: 8281-8296
Published: 2013
doi: https://doi.org/10.1021/jo4013755

23. Antimicrobial Activity of 8-Hydroxyquinoline and Transition Metal Complexes

By: Srisung, S., Suksrichav, T., Prachayasi, S., Ruchirawat, S., and Prachayasi, V.
International Journal of Pharmacology
Vol.: 9
No.:
Page: 170-175
Published: 2013
doi: https://doi.org/10.3923/ijp.2013.170.175

24. Directed biosynthesis through biohalogenation of secondary metabolites of the marine-derived fungus Aspergillus unguis

By: Sureram, S., Kesornpun, C., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
RSC Advances
Vol.: 3
No.: 6
Page: 1781-1788
Published: 2013
doi: https://doi.org/10.1039/C2RA23021F

25. Facile synthesis of diarylmethanes via quinone methides

By: Tangdenpaisal, K., Phakhodee, W., Ruchirawat, S., and Ploypradith, P.
Tetrahedron
Vol.: 69
No.: 2
Page: 933-941
Published: 2013
doi: https://doi.org/10.1016/j.tet.2012.10.087

26. Synthesis of 2,4-unsubstituted quinoline-3-carboxylic acid ethyl esters from arylmethyl azides via a domino process

By: Tummatorn, J., Thongsornkleeb, C., Ruchirawat, S., and Gettongsong, T.
Organic & Biomolecular Chemistry
Vol.: 11
No.: 9
Page: 1463-1467
Published: 2013
doi: https://doi.org/10.1039/c3ob27493d

2012

Updated on September 18, 2020

1. In Vitro Acanthamoebicidal Activity of Fusaric Acid and Dehydrofusaric Acid from an Endophytic Fungus Fusarium sp Tlau3

By: Boonman, N., Prachya, S., Boonmee, A., Kittakoop, P., Wiyakrutta, S., Sriubolmas, N., Warit, S., and Chusattayanond, A. D. A.
Planta Medica
Vol.: 78
No.: 14
Page: 1562-1567
Published: 2012
doi: https://doi.org/10.1055/s-0032-1315146

2. Palladium-catalyzed intramolecular C-H amidation: synthesis and biological activities of indolobenzazocin-8-ones

By: Boonya-udtayan, S., Eno, M., Ruchirawat, S., Mahidol, C., and Thasana, N.
Tetrahedron
Vol.: 68
No.: 50
Page: 10293-10301
Published: 2012
doi: https://doi.org/10.1016/j.tet.2012.10.011

3. Unprecedented furan-2-carbonyl C-glycosides and phenolic diglycosides from Scleropyrum pentandrum

By: Disadee, W., Mahidol, C., Sahakitpichan, P., Sitthimonchai, S., Ruchirawat, S., and Kanchanapoom, T.
Phytochemistry
Vol.: 74
No.:
Page: 115-122
Published: 2012
doi: https://doi.org/10.1016/j.phytochem.2011.11.001

4. 5-Formylfurfuryl esters from Duabanga grandiflora

By: Kaweetripob, W., Mahidol, C., Prachyawarakorn, V., Prawat, H., and Ruchirawat, S.
Phytochemistry
Vol.: 76
No.:
Page: 78-82
Published: 2012
doi: https://doi.org/10.1016/j.phytochem.2012.01.014

5. BIOACTIVE COMPOUNDS FROM THAI MARINE-DERIVED FUNGI

By: Kittakoop, P.
Pharmaceutical Biology
Vol.: 50
No.: 5
Page: 650-650
Published: 2012
doi:

6. NATURAL PRODUCTS WITH BIOLOGICAL ACTIVITIES FROM THAI BIORESOURCES

By: Mahidol, C.
Pharmaceutical Biology
Vol.: 50
No.: 5
Page: 611-611
Published: 2012
doi:

7. Nitrone formation in phosphate buffer and aqueous solutions: novel chemistry inspired by a natural product

By: Pansanit, A., Ingavat, N., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Tetrahedron Letters
Vol.: 53
No.: 16
Page: 2129-2131
Published: 2012
doi: https://doi.org/10.1016/j.tetlet.2012.02.046

8. Synthesis and cytotoxicity of novel 2,2′-bis- and 2,2′,2″-tris-indolylmethanes-based bengacarboline analogs

By: Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Archives of pharmacal research
Vol.: 35
No.: 6
Page: 949-954
Published: 2012
doi: https://doi.org/10.1007/s12272-012-0601-1

9. Synthesis and cytotoxicity of novel 2,2 ‘-bis- and 2,2 ‘,2 ” Euro(3)-tris-indolylmethanes-based bengacarboline analogs

By: Pingaew, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Archives of Pharmacal Research
Vol.: 35
No.: 6
Page: 949-954
Published: 2012
doi: https://doi.org/10.1007/s12272-012-0601-1

10. Chemical Constituents and Antioxidant Activity of Hydnophytum formicarum Jack

By: Prachayasittikul, S., Pingaew, R., Yarnkamon, V., Worachartcheewan, A., Wanwimolruk, S., Ruchirawat, S., and Prachayasittikul, V.
International Journal of Pharmacology
Vol.: 8
No.: 5
Page: 440-444
Published: 2012
doi: https://doi.org/10.3923/ijp.2012.440.444

11. Metal Complexes of Uracil Derivatives with Cytotoxicity and Superoxide Scavenging Activity

By: Prachayasittikul, S., Worachartcheewan, A., Pingaew, R., Suksrichavalit, T., Isarankura-Na-Ayudhya, C., Ruchirawat, S., and Prachayasittikul, V.
Letters in Drug Design & Discovery
Vol.: 9
No.: 3
Page: 282-287
Published: 2012
doi: https://doi.org/10.2174/157018012799129918

12. Antioxidant and antimicrobial activities of Saraca thaipingensis Cantley ex Prain

By: Prachayasittikul, S., Worachartcheewan, A., Yainoy, S., Lomchoey, N., Kittiphatcharin, P., Ruchirawat, S., and Prachayasittikul, V.
Asian Pacific Journal of Tropical Biomedicine
Vol.: 2
No.: 2, Supplement
Page: S796-S799
Published: 2012
doi: https://doi.org/10.1016/S2221-1691

13. Iodo-sesquiterpene hydroquinone and brominated indole alkaloids from the Thai sponge Smenospongia sp

By: Prawat, H., Mahidol, C., Kaweetripob, W., Wittayalai, S., and Ruchirawat, S.
Tetrahedron
Vol.: 68
No.: 34
Page: 6881-6886
Published: 2012
doi: https://doi.org/10.1016/j.tet.2012.06.018

14. Adaptogenic-active components from Kaempferia parviflora rhizomes

By: Pripdeevech, P., Pitija, K., Rujjanawate, C., Pojanagaroon, S., Kittakoop, P., and Wongpornchai, S.
Food Chemistry
Vol.: 132
No.: 3
Page: 1150-1155
Published: 2012
doi: https://doi.org/10.1016/j.foodchem.2011.11.025

15. A novel tricyclic polyketide and its biosynthetic precursor azaphilone derivatives from the endophytic fungus Dothideomycete sp

By: Senadeera, S. P. D., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Organic & Biomolecular Chemistry
Vol.: 10
No.: 35
Page: 7220-7226
Published: 2012
doi: https://doi.org/10.1039/c2ob25959a

16. Antimycobacterial activity of bisbenzylisoquinoline alkaloids from Tiliacora triandra against multidrug-resistant isolates of Mycobacterium tuberculosis

By: Sureram, S., Senadeera, S. P. D., Hongmanee, P., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Bioorganic and Medicinal Chemistry Letters
Vol.: 22
No.: 8
Page: 2902-2905
Published: 2012
doi: https://doi.org/10.1016/j.bmcl.2012.02.053

17. Depsidones, Aromatase Inhibitors and Radical Scavenging Agents from the Marine-Derived Fungus Aspergillus unguis CRI282-03

By: Sureram, S., Wiyakrutta, S., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Planta Medica
Vol.: 78
No.: 6
Page: 582-588
Published: 2012
doi: https://doi.org/10.1055/s-0031-1298228

18. Acid-promoted rearrangement of arylmethyl azides: applications toward the synthesis of N-arylmethyl arenes and polycyclic heteroaromatic compounds

By: Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
Tetrahedron
Vol.: 68
No.: 24
Page: 4732-4739
Published: 2012
doi: https://doi.org/10.1016/j.tet.2012.04.014

19. Lycophlegmariols A-D: Cytotoxic serratene triterpenoids from the club moss Lycopodium phlegrnaria L

By: Wittayalai, S., Sathalalai, S., Thorroad, S., Worawittayanon, P., Ruchirawat, S., and Thasana, N.
Phytochemistry
Vol.: 76
No.:
Page: 117-123
Published: 2012
doi: https://doi.org/10.1016/j.phytochem.2012.01.006

20. Antioxidant, cytotoxicity, and QSAR study of 1-adamantylthio derivatives of 3-picoline and phenylpyridines

By: Worachartcheewan, A., Prachayasittikul, S., Pingaew, R., Nantasenamat, C., Tantimongcolwat, T., Ruchirawat, S., and Prachayasittikul, V.
Medicinal Chemistry Research
Vol.: 21
No.: 11
Page: 3514-3522
Published: 2012
doi: https://doi.org/10.1007/s00044-011-9903-y

21. Iridoid and flavone glycosides from Asystasia gangetica subsp micrantha and Asystasia salicifolia and their antioxidant activities

By: Worawittayanon, P., Ruadreo, J., Disadee, W., Sahakitpichan, P., Sitthimonchai, S., Thasana, N., Ruchirawat, S., and Kanchanapoom, T.
Biochemical Systematics and Ecology
Vol.: 40
No.:
Page: 38-42
Published: 2012
doi: https://doi.org/10.1016/j.bse.2011.08.016

22. Synthesis of benzoindoloquinolizines via a Cu(I)-mediated C-N bond formation

By: Worayuthakarn, R., Nealmongkol, P., Ruchirawat, S., and Thasana, N.
Tetrahedron
Vol.: 68
No.: 13
Page: 2864-2875
Published: 2012
doi: https://doi.org/10.1016/j.tet.2012.01.094

2011

Updated on September 18, 2020

1. Itaconic acid derivatives and diketopiperazine from the marine-derived fungus Aspergillus aculeatus CRI322-03

By: Antia, B. S., Aree, T., Kasettrathat, C., Wiyakrutta, S., Ekpa, O. D., Ekpe, U. J., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 72
No.: 8
Page: 816-820
Published: 2011
doi: https://doi.org/10.1016/j.phytochem.2011.02.013

2. Hybrid flavan-chalcones, aromatase and lipoxygenase inhibitors, from Desmos cochinchinensis

By: Bajgai, S. P., Prachyawarakorn, V., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 72
No.: 16
Page: 2062-2067
Published: 2011
doi: https://doi.org/10.1016/j.phytochem.2011.07.002

3. A simple microwave-assisted preparation of 2-bromo-1-alkenes from 1-alkynes using the LiBr-TMSCl-TEAB reagent system

By: Bunrit, A., Ruchirawat, S., and Thongsornkleeb, C.
Tetrahedron Letters
Vol.: 52
No.: 24
Page: 3124-3127
Published: 2011
doi: https://doi.org/10.1016/j.tetlet.2011.04.025

4. Flavonol 3-O-robinobiosides and 3-O-(2 ”-O-alpha-rhamnopyranosyl)-robinobiosides from Sesuvium portulacastrum

By: Disadee, W., Mahidol, C., Sahakitpichan, P., Sitthimonchai, S., Ruchirawat, S., and Kanchanapoom, T.
Tetrahedron
Vol.: 67
No.: 23
Page: 4221-4226
Published: 2011
doi: https://doi.org/10.1016/j.tet.2011.04.041

5. A novel approach for the synthesis of lophocladines A, B and C1 analogues

By: Disadee, W., Ploypradith, P., Aree, T., Chaichit, N., and Ruchirawat, S.
Tetrahedron Letters
Vol.: 52
No.: 46
Page: 6142-6144
Published: 2011
doi: https://doi.org/10.1016/j.tetlet.2011.09.032

6. INVESTIGATION ON BIOLOGICAL ACTIVITIES OF ANTHRANILIC ACID SULFONAMIDE ANALOGS

By: Doungsoongnuen, S., Worachartcheewan, A., Pingaew, R., Suksrichavalit, T., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 10
No.:
Page: 155-161
Published: 2011
doi:

7. Molecular dynamics investigation of psalmopeotoxin I. Probing the relationship between 3D structure, anti-malarial activity and thermal stability

By: Gleeson, M. P., Deechongkit, S., and Ruchirawat, S.
Journal of Molecular Modeling
Vol.: 17
No.: 4
Page: 769-775
Published: 2011
doi: https://doi.org/10.1007/s00894-010-0732-6

8. Biological Activities of Synthetic Oligosaccharides and Glycolipids from Mycobacteria

By: Hutacharoen, P., Ruchirawat, S., and Boonyarattanakalin, S.
Journal of Carbohydrate Chemistry
Vol.: 30
No.: 7-9
Page: 415-437
Published: 2011
doi: https://doi.org/10.1080/07328303.2011.621041

9. Asperaculin A, a Sesquiterpenoid from a Marine-Derived Fungus, Aspergillus aculeatus

By: Ingavat, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Journal of Natural Products
Vol.: 74
No.: 7
Page: 1650-1652
Published: 2011
doi: https://doi.org/10.1021/np200221w

10. Overcoming Multidrug Resistance in Human Lung Cancer with Novel Benzo a quinolizin-4-ones

By: Kanintronkul, Y., Worayuthakarn, R., Thasana, N., Winayanuwattikun, P., Pattanapanyasat, K., Surarit, R., Ruchirawat, S., and Svasti, J.
Anticancer Research
Vol.: 31
No.: 3
Page: 921-927
Published: 2011
doi:

11. Protoberberine Alkaloids and Cancer Chemopreventive Properties of Compounds from Alangium salviifolium

By: Pailee, P., Prachyawarakorn, V., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
European Journal of Organic Chemistry
Vol.: 2011
No.: 20-21
Page: 3809-3814
Published: 2011
doi: https://doi.org/10.1002/ejoc.201100423

12. Antiplasmodial and antimycobacterial cyclopeptide alkaloids from the root of Ziziphus mauritiana

By: Panseeta, P., Lomchoey, K., Prabpai, S., Kongsaeree, P., Suksamrarn, A., Ruchirawat, S., and Suksamrarn, S.
Phytochemistry
Vol.: 72
No.: 9
Page: 909-915
Published: 2011
doi: https://doi.org/10.1016/j.phytochem.2011.03.003

13. Synthesis and structure-activity relationship of 2-thiopyrimidine-4-one analogs as antimicrobial and anticancer agents

By: Prachayasittikul, S., Worachartcheewan, A., Nantasenamat, C., Chinworrungsee, M., Sornsongkhram, N., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Medicinal Chemistry
Vol.: 46
No.: 2
Page: 738-742
Published: 2011
doi: https://doi.org/10.1016/j.ejmech.2010.12.009

14. Longeracemosones A-F, Aromatase Inhibitors from Dunbaria longeracemosa

By: Prachyawarakorn, V., Mahidol, C., and Ruchirawat, S.
European Journal of Organic Chemistry
Vol.: 2011
No.: 20-21
Page: 3803-3808
Published: 2011
doi: https://doi.org/10.1002/ejoc.201100410

15. Nitrogenous sesquiterpenes from the Thai marine sponge Halichondria sp

By: Prawat, H., Mahidol, C., Wittayalai, S., Intachote, P., Kanchanapoom, T., and Ruchirawat, S.
Tetrahedron
Vol.: 67
No.: 31
Page: 5651-5655
Published: 2011
doi: https://doi.org/10.1016/j.tet.2011.05.094

16. PEG-b-PCL and PEG-b-PLA polymeric micelles as nanocarrieres for lamellarin N delivery

By: Pungkham, H., Swatdipakdi, N., Theerasilp, M., Karnkla, S., Chittchang, M., Ploypradith, P., and Nasongkla, N.
Conference proceedings: Annual International Conference of the IEEE Engineering in Medicine and Biology Society. IEEE Engineering in Medicine and Biology Society. Annual Conference
Vol.: 2011
No.:
Page: 3245-3248
Published: 2011
doi: https://doi.org/10.1109/iembs.2011.6090882

17. Pt(IV)-catalyzed generation and 4+2 -cycloaddition reactions of o-quinone methides

By: Radomkit, S., Sarnpitak, P., Tummatorn, J., Batsomboon, P., Ruchirawat, S., and Ploypradith, P.
Tetrahedron
Vol.: 67
No.: 21
Page: 3904-3914
Published: 2011
doi: https://doi.org/10.1016/j.tet.2011.03.059

18. 3-Hydroxydihydrobenzofuran Glucosides from Gnaphalium polycaulon

By: Sahakitpichan, P., Disadee, W., Ruchirawat, S., and Kanchanapoom, T.
Chemical & Pharmaceutical Bulletin
Vol.: 59
No.: 9
Page: 1160-1162
Published: 2011
doi: https://doi.org/10.1248/cpb.59.1160

19. Unusual glycosides of pyrrole alkaloid and 4 ‘-hydroxyphenylethanamide from leaves of Moringa oleifera

By: Sahakitpichan, P., Mahidol, C., Disadee, W., Ruchirawat, S., and Kanchanapoom, T.
Phytochemistry
Vol.: 72
No.: 8
Page: 791-795
Published: 2011
doi: https://doi.org/10.1016/j.phytochem.2011.02.021

20. Exploring the molecular basis for selective cytotoxicity of lamellarins against human hormone-dependent T47D and hormone-independent MDA-MB-231 breast cancer cells

By: Thipnate, P., Chittchang, M., Thasana, N., Saparpakorn, P., Ploypradith, P., and Hannongbua, S.
Monatshefte fur Chemie
Vol.: 142
No.: 1
Page: 97-109
Published: 2011
doi: https://doi.org/10.1007/s00706-010-0409-y

21. Radical Scavenging and Antioxidant Activities of Isocoumarins and a Phthalide from the Endophytic Fungus Colletotrichum sp

By: Tianpanich, K., Prachya, S., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Journal of Natural Products
Vol.: 74
No.: 1
Page: 79-81
Published: 2011
doi: https://doi.org/10.1021/np1003752

22. BIOACTIVE 4-HYDROXYCINNAMIDE AND BIOACTIVITIES OF POLYALTHIA CERASOIDES

By: Treeratanapiboon, L., Worachartcheewan, A., Suksrichavalit, T., Kiatfuengfoo, R., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 10
No.:
Page: 16-22
Published: 2011
doi:

2010

Updated on September 18, 2020

1. Alpha-glucosidase inhibitory, aromatase inhibitory, and antiplasmodial activities of a biflavonoid GB1 from Garcinia kola stem bark

By: Antia, B. S., Pansanit, A., Ekpa, O. D., Ekpe, U. J., Mahidol, C., and Kittakoop, P.
Planta Medica
Vol.: 76
No.: 3
Page: 276-277
Published: 2010
doi: https://doi.org/10.1055/s-0029-1186081

2. Paraherquamide E

By: Aree, T., Antia, B. S., Ekpa, O. D., and Kittakoop, P.
Acta Crystallographica Section E
Vol.: 66
No.: 9
Page: o2227
Published: 2010
doi: https://doi.org/10.1107/S1600536810030795

3. Synthesis and biological activities of azalamellarins

By: Boonya-Udtayan, S., Yotapan, N., Woo, C., Bruns, C. J., Ruchirawat, S., and Thasana, N.
Chemistry, an Asian Journal
Vol.: 5
No.: 9
Page: 2113-2123
Published: 2010
doi: https://doi.org/10.1002/asia.201000237

4. Part 1: Antiplasmodial, Cytotoxic, Radical Scavenging and Antioxidant Activities of Thai Plants in the Family Acanthaceae

By: Charoenchai, P., Vajrodaya, S., Somprasong, W., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Planta Medica
Vol.: 76
No.:
Page: 1940-1943
Published: 2010
doi: https://doi.org/10.1055/s-0030-1250045

5. Assessing the drug-likeness of lamellarins, a marine-derived natural product class with diverse oncological activities

By: Chittchang, M., Paul Gleeson, M., Ploypradith, P., and Ruchirawat, S.
European Journal of Medicinal Chemistry
Vol.: 45
No.: 6
Page: 2165-2172
Published: 2010
doi: https://doi.org/10.1016/j.ejmech.2010.01.053

6. Curvularides A-E: antifungal hybrid peptide-polyketides from the endophytic fungus Curvularia geniculata

By: Chomcheon, P., Wiyakrutta, S., Aree, T., Sriubolmas, N., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Chemistry
Vol.: 16
No.: 36
Page: 11178-11185
Published: 2010
doi: https://doi.org/10.1002/chem.201000652

7. Synthesis, biophysical, and biological studies of wild-type and mutant psalmopeotoxins—Anti-malarial cysteine knot peptides from Psalmopoeus cambridgei

By: Kamolkijkarn, P., Prasertdee, T., Netirojjanakul, C., Sarnpitak, P., Ruchirawat, S., and Deechongkit, S.
Peptides
Vol.: 31
No.: 4
Page: 533-540
Published: 2010
doi: https://doi.org/10.1016/j.peptides.2010.01.001

8. Acanmontanoside, a new phenylethanoid diglycoside from Acanthus montanus

By: Noiarsa, P., Ruchirawat, S., and Kanchanapoom, T.
Molecules
Vol.: 15
No.: 12
Page: 8967-8972
Published: 2010
doi: https://doi.org/10.3390/molecules15128967

9. Glutarimide Alkaloids and a Terpenoid Benzoquinone from Cordia globifera

By: Parks, J., Gyeltshen, T., Prachyawarakorn, V., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Journal of Natural Products
Vol.: 73
No.: 5
Page: 992-994
Published: 2010
doi: https://doi.org/10.1021/np100078s

10. Synthesis, Cytotoxic and Antimalarial Activities of Benzoyl Thiosemicarbazone Analogs of Isoquinoline and Related Compounds

By: Pingaew, R., Prachayasittikul, S., and Ruchirawat, S.
Molecules (Basel, Switzerland)
Vol.: 15
No.:
Page: 988-996
Published: 2010
doi: https://doi.org/10.3390/molecules15020988

11. A new sulfoxide analog of 1,2,3,6-tetrahydrophenylpyridine and antimicrobial activity

By: Prachayasittikul, S., Pingaew, R., Worachartcheewan, A., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 9
No.:
Page: 102
Published: 2010
doi: https://doi.org/10.17877/DE290R-15807

12. New bioactive triterpenoids and antimalarial activity of Diospyros rubra Lec

By: Prachayasittikul, S., Saraban, P., Cherdtrakulkiat, R., Ruchirawat, S., and Prachayasittikul, V.
EXCLI journal
Vol.: 9
No.:
Page: 1-10
Published: 2010
doi:

13. Elucidating the structure-activity relationships of the vasorelaxation and antioxidation properties of thionicotinic acid derivatives

By: Prachayasittikul, S., Wongsawatkul, O., Worachartcheewan, A., Nantasenamat, C., Ruchirawat, S., and Prachayasittikul, V.
Molecules
Vol.: 15
No.: 1
Page: 198-214
Published: 2010
doi: https://doi.org/10.3390/molecules15010198

14. Vasorelaxation and Superoxide Scavenging Activities of Orotic Acid

By: Prachayasittikul, S., Wongsawatkul, O., Worachartcheewan, A., Ruchirawat, S., and Prachayasittikul, V.
International Journal of Pharmacology
Vol.: 6
No.:
Page:
Published: 2010
doi: https://doi.org/10.3923/ijp.2010.413.418

15. Bacillus subtilis SSE4 produces subtulene A, a new lipopeptide antibiotic possessing an unusual C15 unsaturated beta-amino acid

By: Thasana, N., Prapagdee, B., Rangkadilok, N., Sallabhan, R., Aye, S. L., Ruchirawat, S., and Loprasert, S.
FEBS Letters
Vol.: 584
No.: 14
Page: 3209-3214
Published: 2010
doi: https://doi.org/10.1016/j.febslet.2010.06.005

16. A Convergent General Strategy for the Functionalized 2-Aryl Cycloalkyl-Fused Chromans: Intramolecular Hetero-Diels–Alder Reactions of ortho-Quinone Methides

By: Tummatorn, J., Ruchirawat, S., and Ploypradith, P.
Chemistry – A European Journal
Vol.: 16
No.: 5
Page: 1445-1448
Published: 2010
doi: https://doi.org/10.1002/chem.200902403

17. Polymerization of mannosyl tricyclic orthoesters for the synthesis of alpha(1-6) mannopyranan-the backbone of lipomannan

By: Yongyat, C., Ruchirawat, S., and Boonyarattanakalin, S.
Bioorg Med Chem
Vol.: 18
No.: 11
Page: 3726-3734
Published: 2010
doi: https://doi.org/10.1016/j.bmc.2010.04.014

2009

Updated on September 18, 2020

1. (E)-2,4,7-Trichloro-3-hydroxy-8-methoxy-1,9-dimethyl-6-(1-methyl-1-propenyl)-11H-dibenzo[b,e][1,4]dioxepin-11-one monohydrate (nidulin monohydrate)

By: Aree, T., Sanya, S., Ngamrojanavanich, N., and Kittakoop, P.
Acta Crystallographica Section E
Vol.: 65
No.:
Page:
Published: 2009
doi: https://doi.org/10.1107/S1600536809036277/sj2646Isup2.hkl

2. Generation of ortho-quinone methides by p-TsOH on silica and their hetero-Diels-Alder reactions with styrenes

By: Batsomboon, P., Phakhodee, W., Ruchirawat, S., and Ploypradith, P.
Journal of Organic Chemistry
Vol.: 74
No.: 10
Page: 4009-4012
Published: 2009
doi: https://doi.org/10.1021/jo900504y

3. Cytotoxicities and Structure–Activity Relationships of Natural and Unnatural Lamellarins toward Cancer Cell Lines

By: Chittchang, M., Batsomboon, P., Ruchirawat, S., and Ploypradith, P.
ChemMedChem
Vol.: 4
No.: 3
Page: 457-465
Published: 2009
doi: https://doi.org/10.1002/cmdc.200800339

4. Aromatase inhibitory, radical scavenging, and antioxidant activities of depsidones and diaryl ethers from the endophytic fungus Corynespora cassiicola L36

By: Chomcheon, P., Wiyakrutta, S., Sriubolmas, N., Ngamrojanavanich, N., Kengtong, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 70
No.: 3
Page: 407-413
Published: 2009
doi: https://doi.org/10.1016/j.phytochem.2009.01.007

5. Metabolites from the endophytic mitosporic Dothideomycete sp. LRUB20

By: Chomcheon, P., Wiyakrutta, S., Sriubolmas, N., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 70
No.: 1
Page: 121-127
Published: 2009
doi: https://doi.org/10.1016/j.phytochem.2008.10.007

6. Biomimetic Transformation and Biological Activities of Globiferin, a Terpenoid Benzoquinone from Cordia globifera

By: Dettrakul, S., Surerum, S., Rajviroongit, S., and Kittakoop, P.
Journal of Natural Products
Vol.: 72
No.: 5
Page: 861-865
Published: 2009
doi: https://doi.org/10.1021/np9000703

7. Aspergillusol A, an alpha-glucosidase inhibitor from the marine-derived fungus Aspergillus aculeatus

By: Ingavat, N., Dobereiner, J., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Journal of Natural Products
Vol.: 72
No.: 11
Page: 2049-2052
Published: 2009
doi: https://doi.org/10.1021/np9003883

8. Bioactive Scalaranes from the Thai Sponge Hyrtios gumminae

By: Mahidol, C., Prawat, H., Sangpetsiripan, S., and Ruchirawat, S.
Journal of Natural Products
Vol.: 72
No.: 10
Page: 1870-1874
Published: 2009
doi: https://doi.org/10.1021/np900267v

9. A new synthetic approach towards isoquinobenzazepinone and isoindolinobenzazepinone using acid-mediated cyclisation and Heck reaction

By: Phakhodee, W., Ploypradith, P., Sahakitpichan, P., and Ruchirawat, S.
Tetrahedron
Vol.: 65
No.: 1
Page: 351-356
Published: 2009
doi: https://doi.org/10.1016/j.tet.2008.10.044

10. Isolation of Bioactive Metabolites from Root Extracts of Polyalthia Debilis

By: Prachayasittikul, S., Buttrawong, K., Worachartcheewan, A., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Scientific Research ISSN
Vol.: 38
No.:
Page: 1450-1216
Published: 2009
doi:

11. Bioactive Azafluorenone Alkaloids from Polyalthia debilis (Pierre) Finet & Gagnep

By: Prachayasittikul, S., Manam, P., Chinworrungsee, M., Isarankura-Na-Ayudhya, C., Ruchirawat, S., and Prachayasittikul, V.
Molecules (Basel, Switzerland)
Vol.: 14
No.:
Page: 4414-4424
Published: 2009
doi: https://doi.org/10.3390/molecules14114414

12. Synthesis and Novel Bioactivities of Substituted 6-Propylthiouracils

By: Prachayasittikul, S., Sornsongkhram, N., Pingaew, R., Techatanachai, S., Ruchirawat, S., and Prachayasittikul, V.
European Journal of Scientific Research
Vol.: 36
No.:
Page: 236
Published: 2009
doi:

13. Factors affecting orthogonality in the deprotection of 2,4-di-protected aromatic ethers employing solid-supported acids

By: Tangdenpaisal, K., Sualek, S., Ruchirawat, S., and Ploypradith, P.
Tetrahedron
Vol.: 65
No.: 22
Page: 4316-4325
Published: 2009
doi: https://doi.org/10.1016/j.tet.2009.03.089

2008

Updated on September 18, 2020

1. Cytotoxic and antiplasmodial substances from marine-derived fungi, Nodulisporium sp and CRI247-01

By: Kasettrathat, C., Ngamrojanavanich, N., Wiyakrutta, S., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Phytochemistry
Vol.: 69
No.: 14
Page: 2621-2626
Published: 2008
doi: https://doi.org/10.1016/j.phytochem.2008.08.005

2. Investigation of the acid-mediated cyclisation of amide acetal for the synthesis of benzazepinone

By: Phakhodee, W., Sahakitpichan, P., Deechongkit, S., and Ruchirawat, S.
Heterocycles
Vol.: 75
No.: 8
Page: 1963-1970
Published: 2008
doi:

3. Diketopiperazines and phthalides from a marine derived fungus of the order pleosporales

By: Prachyawarakorn, V., Mahidol, C., Sureram, S., Sangpetsiripan, S., Wiyakrutta, S., Ruchirawat, S., and Kittakoop, P.
Planta Medica
Vol.: 74
No.: 1
Page: 69-72
Published: 2008
doi: https://doi.org/10.1055/s-2007-993783

4. A facile synthesis of telisatin a via microwave-promoted annulation and Reformatsky reaction

By: Thasana, N., Bjerke-Kroll, B., and Ruchirawat, S.
Synlett
Vol.:
No.: 4
Page: 505-508
Published: 2008
doi: https://doi.org/10.1055/s-2008-1042764

5. Synthesis of unsymmetrical benzil licoagrodione

By: Worayuthakarn, R., Boonya-Udtayan, S., Arom-Oon, E., Ploypradith, P., Ruchirawat, S., and Thasana, N.
Journal of Organic Chemistry
Vol.: 73
No.: 18
Page: 7432-7435
Published: 2008
doi: https://doi.org/10.1021/jo8013353

2007

Updated on September 18, 2020

1. Application of the hypervalent iodine reagent to the synthesis of some pentasubstituted aporphine alkaloids

By: Pingaew, R., and Ruchirawat, S.
Synlett
Vol.:
No.: 15
Page: 2363-2366
Published: 2007
doi: https://doi.org/10.1055/s-2007-985596

2. Cytotoxic mycoepoxydiene derivatives from an endophytic fungus Phomopsis sp isolated from Hydnocarpus anthelminthicus

By: Prachya, S., Wiyakrutta, S., Sriubolmas, N., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Planta Medica
Vol.: 73
No.: 13
Page: 1418-1420
Published: 2007
doi: https://doi.org/10.1055/s-2007-990240

3. The Asian CORE Program: Cutting-Edge Organic Chemistry in Asia

By: Ruchirawat, S., Chittchang, M., and Ploypradith, P.
ScienceAsia
Vol.: 33(s1)
No.:
Page:
Published: 2007
doi: https://doi.org/10.2306/scienceasia1513-1874.2007.33(s1).029

4. Copper(I)-mediated and microwave-assisted C-aryl-O-carboxylic coupling: Synthesis of benzopyranones and isolamellarin alkaloids

By: Thasana, N., Worayuthakarn, R., Kradanrat, P., Hohn, E., Young, L. R., and Ruchirawat, S.
Journal of Organic Chemistry
Vol.: 72
No.: 24
Page: 9379-9382
Published: 2007
doi: https://doi.org/10.1021/jo701599g

5. Diterpenoids from the roots of Croton oblongifolius

By: Youngsa-Ad, W., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., Prawat, H., and Kittakoop, P.
Planta Medica
Vol.: 73
No.: 14
Page: 1491-1494
Published: 2007
doi: https://doi.org/10.1055/s-2007-990247

Research

Publications

RESEARCH IN CHEMICAL SCIENCES (CS)

2024

4-Aryl-1H-isochromenes Synthesis from Triol Derivatives through Brønsted Acid-Catalyzed Pinacol Rearrangement/Intramolecular Cyclization Sequence

Albiflorenes A–L, polyoxygenated cyclohex(a/e)ne diterpene esters from Kaempferia albiflora

Altenusin, a fungal metabolite, alleviates TGF-β1-induced EMT in renal proximal tubular cells and renal fibrosis in unilateral ureteral obstruction

Breast Cancer Prevention by Dietary Polyphenols: Microemulsion Formulation and In Vitro Studies

Cascade Cyclization of o-(2-Acyl-1-ethynyl)benzaldehydes with Amino Acid Derivatives: Synthesis of Indeno[2,1-c]pyran-3-ones and 1-Oxazolonylisobenzofurans via the Erlenmeyer-Plöchl Azlactone Reaction

Chemical constituents from Microstachys chamaelea (Euphorbiaceae) with cytotoxic and antioxidant properties

Controllable Chemoselectivity Cascade Reactions for the Synthesis of Phenanthrenols via Palladium-Catalyzed-Suzuki/Heck Reaction and Michael Addition

Cytotoxic stress caused by azalamellarin D (AzaD) interferes with cellular protein translation by targeting the nutrient-sensing kinase mTOR

Dihydro-10H-indeno[1,2-b]benzofurans and Tetrahydroindeno[1,2-c]isochromenes via Stereoselective Intramolecular Carbocation Cascade Cyclization

Diphenyl ethers from the cultured lichen mycobiont of Graphis handelii Zahlbr

Discovery of procyanidin condensed tannins of (−)-epicatechin from Kratom, Mitragyna speciosa, as virucidal agents against SARS-CoV-21

Effects of barakol from Cassia siamea on neuroblastoma SH-SY5Y cell line: A potential combined therapy with doxorubicin

Electron Donor-Acceptor Complex-Enabled Autoinductive Conversion of Acylnitromethanes to Acylnitrile Oxides in a Photochemical Machetti-De Sarlo Reaction: Synthesis of 5-Substituted 3-Acylisoxazoles

Enantioselective Reductive Cyclization of Alkynyl-Tethered Cyclohexadienones Catalyzed by Rhodium Complexes

Evolution-guided engineering of trans-acyltransferase polyketide synthases

Facile metabolic reprogramming distinguishes mycobacterial adaptation to hypoxia and starvation: ketosis drives starvation-induced persistence in M. bovis BCG

Grewiifopenes A–K, bioactive clerodane diterpenoids from Casearia grewiifolia Vent

Huperzine A Regulates the Physiological Homeostasis of Amyloid Precursor Protein Proteolysis and Tau Protein Conformation—A Computational and Experimental Investigation

Inhibition of Giardia duodenalis by isocryptolepine -triazole adducts and derivatives

Ligand-Based Virtual Screening for Discovery of Indole Derivatives as Potent DNA Gyrase ATPase Inhibitors Active against Mycobacterium tuberculosis and Hit Validation by Biological Assays

Metal- and photocatalyst-free approach to visible-light-induced acylation of quinoxalinones

Molecular Reconstruction with Stereochemical Relay: An Investigation into the Rearrangement of Spiro[4.5]decadienone to Benzoxepane

Novel naphthoquinones as potent aromatase inhibitors: Synthesis, anticancer, and in silico studies

Pharmacological Properties of White Mulberry (Morus alba L.) Leaves: Suppressing Migratory and Invasive Activities Against A549 Lung Cancer Cells

Rapid and Scalable Production of Functional SARS-CoV-2 Virus-like Particles (VLPs) by a Stable HEK293 Cell Pool

A structure-based virtual high-throughput screening, molecular docking, molecular dynamics and MM/PBSA study identified novel putative drug-like dual inhibitors of trypanosomal cruzain and rhodesain cysteine proteases

Sultines as o -Quinodimethane Precursors in an Oxa-Diels-Alder Reaction: Synthesis of Functionalized Isochromans

Synthesis, Antiacetylcholinesterase Activity, and Molecular Dynamics Simulation of Aporphine-benzylpyridinium Conjugates

Synthesis, in silico, in vitro evaluation of furanyl- and thiophenyl-3-phenyl-1H-indole-2-carbohydrazide derivatives as tubulin inhibitors and anticancer agents

A toluidine blue/porous organic polymer/2D MoSe2 nanocomposite as an electrochemical signaling platform for a sensitive label-free aflatoxin B1 bioassay in some crops

Two Cytochrome P450 Enzymes Form the Tricyclic Nested Skeleton of Meroterpenoids by Sequential Oxidative Reactions

Two new serratene triterpenes from club moss cultivars

Unveiling Route for the Synthesis of Tröger’s Bases Through Azide Rearrangement

Vernonia amygdalina Leaf Extract Induces Apoptosis in HeLa Cells: A Metabolomics and Proteomics Study

Visible Light-Induced One-Pot Carbonylation of Alkyl Halides with Aryl Formates

2023

Altenusin inhibits epithelial to mesenchymal transition via suppression of TGF-β/MAPK signaling pathway in human renal proximal tubular cells and unilateral ureteral obstruction mice

The amide derivative of anticopalic acid induces non-apoptotic cell death in triple-negative breast cancer cells by inhibiting FAK activation

Aminochalcones Attenuate Neuronal Cell Death under Oxidative Damage via Sirtuin 1 Activity

Anthelmintic efficacy evaluation and mechanism of N-methylbenzo[d]oxazol-2-amine

Anti-Xanthine Oxidase 5′-Hydroxyhericenes A-D from the Edible Mushroom Hericium erinaceus and Structure Revision of 3-[2,3-Dihydroxy-4-(hydroxymethyl)tetrahydrofuran-1-yl]-pyridine-4,5-diol

Base-Mediated and Silver-Catalyzed Divergent Synthesis of Hydroxynaphthalenamides and Phosphorylated Dihydronaphthylamides from Enone-Oxazolones

Bioisosteric Design Identifies Inhibitors of Mycobacterium tuberculosis DNA Gyrase ATPase Activity

Concise Synthesis of 1,4-Dideoxy-1,4-imino- l -arabinitol (LAB) from d -Xylose by Intramolecular Stereospecific Substitution of a Hydroxy Group

Copper-Catalyzed Guanylation by Ring Extension of 4-Hydroxyquinazoline for the Synthesis of Quinazolino[3,2-a]quinazolinones

Cytotoxic Isopimarane Diterpenoids from Kaempferia koratensis Rhizomes

Degradation of Methylene Blue Using Fly Ash as a Heterogeneous Fenton Catalyst

Discovery of N-methylbenzo[d]oxazol-2-amine as new anthelmintic agent through scalable protocol for the synthesis of N-alkylbenzo[d]oxazol-2-amine and N-alkylbenzo[d]thiazol-2-amine derivatives

Discovery of Novel Naphthoquinone-Chalcone Hybrids as Potent FGFR1 Tyrosine Kinase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling

Divergent synthesis of 3,4-dihydro-2H-benzo[h]chromen-2-one and fluorenone derivatives from ortho-alkynylarylketones

Divergent Synthesis of Isochroman-4-ols, 1,3-Dihydroisobenzo­furans, and Tetrahydro-2 H -indeno[2,1- b ]furan-2-ones via Epoxidation/Cyclization Strategy of (E)-(2-Stilbenyl/Styrenyl)methanols

Fabrication, Optimization, and Characterization of Antibacterial Electrospun Shellac Fibers Loaded with Kaempferia parviflora Extract

Halogenative Annulation Reactions of Alkyne-Tethered N – And O -Containing Arenes: Methods for Accessing Aryl-Fused Halogenated N – And O -Heterocycles

In vitro evaluation of the anti-breast cancer properties and gene expression profiles of Thai traditional formulary medicine extracts

Kaemtakols A–D, highly oxidized pimarane diterpenoids with potent anti-inflammatory activity from Kaempferia takensis

A Mechanistically Deceiving Formation of Aryl(1-indanyl)ketones via Acid-Catalyzed Cyclization of ortho-Alkynylarylmethanols

Microwave-assisted commercial copper-catalyzed aerobic oxidative synthesis of AChE quinazolinone inhibitors under solvent free conditions

Mn(OAc)3-Mediated One-Pot Condensation-Oxidative Annulation of 2-Alkynylanilines and 1,3-Ketoesters: Synthesis of 2-Substituted Quinolines

Novel Pd(ii) pincer complexes bearing salicylaldimine-based benzothiazole derivatives: synthesis, structural characterization, DNA/BSA binding, and biological evaluation

Phlegcarines A-C, three Lycopodium alkaloids from Phlegmariurus carinatus (Desv. ex Poir.) Ching

Phukettosides A–E, mono- and bis-iridoid glycosides, from the leaves of Morinda umbellata L

Protein Modification via Nitrile Oxide−Dehydroalanine Cycloaddition: Formation of Isoxazoline Ring on the Protein Backbone

Rapid synthesis of α(1,2)-D-mannans on the surface of Mycobacterium tuberculosis and their nitric oxide-inducing activities

The redox-sensing mechanism of Agrobacterium tumefaciens NieR as a thiol-based oxidation sensor for hypochlorite stress

Schomburginones A‒J, geranylated benzophenones from the leaves of Garcinia schomburgkiana and their cytotoxic and anti-inflammatory activities

Selective electrophilic cyclization of ortho-carbonylarylacetylenols for the synthesis of cyclopenta[a]naphthalenol and 2-phenylnaphthalen-1-ol analogs

Synthesis of Clausena Alkaloids Using Unique Ring Expansion of Dihydroisoquinolines and Their Cholinesterase Inhibitory Activity

Synthesis of Naphtho[2,3-d]oxazoles via Ag(I) Acid-Mediated Oxazole-Benzannulation of ortho-Alkynylamidoarylketones

Three-Component Aza-Diels-Alder Reaction for the Syntheses of Tetrahydroisoquinoline Derivatives

UHPLC-QQQ-MS and RP-HPLC Detection of Bioactive Alizarin and Scopoletin Metabolites from Morinda citrifolia Root Extracts and Their Antitubercular, Antibacterial, and Antioxidant Activities

Virucidal and Antiviral Polyhydroxylated Fatty Alcohols in Avocado Fruit Pulp (Persea americana) of Booth 7 Cultivar¶

2022

4b-Aryltetrahydroindeno[1,2- a ]indenes by Acid-Catalyzed Trans­annular Cyclization of Benzannulated Cyclooctene Alcohols

Acetogenins from the stems of Uvaria micrantha showing antiproliferative effects on HepG2 liver cancer cells

Acid-dependent Divergent Conversion of ortho-Arylcyclopropanecarbonyl Carboxaldehydes for the Synthesis of Furanodibenzocycloheptenes and Dibenzocycloheptenes

Ag(I)-Catalyzed/Acid-Mediated Cascade Cyclization of ortho-Alkynylaryl-1,3-dicarbonyls to Access Arylnaphthalenelactones and Furanonaphthol Libraries via Aryl-Disengagement

Divergent Synthesis of Isochroman-4-ols, 1,3-Dihydroisobenzofurans, and Tetrahydro-2 H -indeno[2,1- b ]furan-2-ones via Epoxidation/Cyclization Strategy of (E)-(2-Stilbenyl/Styrenyl)methanols

4b-Aryltetrahydroindeno[1,2- a ]indenes by Acid-Catalyzed Transannular Cyclization of Benzannulated Cyclooctene Alcohols

Copper-Mediated C-O/C-N Bond Formation: A Facile Synthesis of 3-Amidocoumarin, 3-Amidoazacoumarin, and N -Aroylindole Derivatives